Celine Valant
Monash University
H-index: 32
Oceania-Australia
Top articles of Celine Valant
Positive allosteric modulation of a GPCR ternary complex
bioRxiv
2024
Celine Valant
H-Index: 20
Arthur Christopoulos
H-Index: 62
Role of conserved tyrosine lid residues in the activation of the M2 muscarinic acetylcholine receptor
Molecular Pharmacology
2023/9/1
Structural basis of efficacy-driven ligand selectivity at GPCRs
Nature Chemical Biology
2023/7
Pharmacological hallmarks of allostery at the M4 muscarinic receptor elucidated through structure and dynamics
Elife
2023/5/30
Acetylcholine receptors (muscarinic) in GtoPdb v. 2023.1
IUPHAR/BPS Guide to Pharmacology CITE
2023/4/26
Importance of receptor expression in the classification of novel ligands at the M2 muscarinic acetylcholine receptor
British Journal of Pharmacology
2023/1/20
Structure–activity relationship of pyrazol-4-yl-pyridine derivatives and identification of a radiofluorinated probe for imaging the muscarinic acetylcholine receptor M4
Acta Pharmaceutica Sinica B
2023/1/1
Ligand-directed biased agonism at human histamine H3 receptor isoforms across Gαi/o-and β-arrestin2-mediated pathways
Biochemical Pharmacology
2023/12/28
Design, synthesis and evaluation of novel 2-phenyl-3-(1H-pyrazol-4-yl) pyridine positive allosteric modulators for the M4 mAChR
European Journal of Medicinal Chemistry
2023/10/5
Emma T Van Der Westhuizen
H-Index: 14
Yao Lu
H-Index: 4
Arthur Christopoulos
H-Index: 62
Celine Valant
H-Index: 20
The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors
British journal of pharmacology
2023/10
Arthur Christopoulos
H-Index: 62
George Abraham
H-Index: 3
Geoffrey Burnstock
H-Index: 68
Stefania Ceruti
H-Index: 24
Nan Chiang
H-Index: 47
Olivier Civelli
H-Index: 40
Steven D Douglas
H-Index: 6
Michael L Garelja
H-Index: 6
Karen J Gregory
H-Index: 30
Debbie L Hay
H-Index: 33
Deron Herr
H-Index: 24
Ahsan Husain
H-Index: 24
Pawel Kozielewicz
H-Index: 8
Dan Larhammar
H-Index: 25
Katie Leach
H-Index: 19
Davide Lecca
H-Index: 20
John D Lee
H-Index: 46
Martin C Michel
H-Index: 40
Duuamene Nyimanu
H-Index: 5
Rithwik Ramachandran
H-Index: 22
Gunnar Schulte
H-Index: 31
Stefan Schulz
H-Index: 4
Roger Summers
H-Index: 32
David Thal
H-Index: 14
Xanomeline displays concomitant orthosteric and allosteric binding modes at the M4 mAChR
Nature communications
2023/9/6
Investigating Drivers for M1 Muscarinic Acetylcholine Receptor‐Mediated Adverse Events by M1 Positive Allosteric Modulators
The FASEB Journal
2022/5
P598. Exploring the Molecular Determinants for Functional Selectivity of the Antipsychotic Xanomeline at Muscarinic Acetylcholine Receptors
Biological Psychiatry
2022/5/1
Biased Profile of Xanomeline at the Recombinant Human M4 Muscarinic Acetylcholine Receptor
ACS Chemical Neuroscience
2022/4/5
Emma T Van Der Westhuizen
H-Index: 14
Vi Pham
H-Index: 11
Arthur Christopoulos
H-Index: 62
Celine Valant
H-Index: 20
Positive allosteric modulation of endogenous delta opioid receptor signaling in the enteric nervous system is a potential treatment for gastrointestinal motility disorders
American Journal of Physiology-Gastrointestinal and Liver Physiology
2022/1/1
Therapeutic potential of allosteric modulators for the treatment of gastrointestinal motility disorders
2022/12/24
Celine Valant
H-Index: 20
Arthur Christopoulos
H-Index: 62
Opportunities and challenges for the development of M1 muscarinic receptor positive allosteric modulators in the treatment for neurocognitive deficits
2022/7/1
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ-Opioid Receptor
Journal of Medicinal Chemistry
2022/9/13
Identification and Preclinical Development of a Radiofluorinated Probe for Imaging the Muscarinic Acetylcholine Receptor M4 by Positron Emission Tomography
2022/6/1
Structural features of iperoxo–BQCA muscarinic acetylcholine receptor hybrid ligands determining subtype selectivity and efficacy
ACS Chemical Neuroscience
2021/12/14
Arthur Christopoulos
H-Index: 62
Celine Valant
H-Index: 20