Arthur Christopoulos
Monash University
H-index: 99
Oceania-Australia
Top articles of Arthur Christopoulos
Cryo-EM Structure of the Human Amylin 1 Receptor in Complex with CGRP and Gs Protein
Biochemistry
2024/4/11
Arthur Christopoulos
H-Index: 62
Denise Wootten
H-Index: 31
Positive allosteric modulation of a GPCR ternary complex
bioRxiv
2024
Celine Valant
H-Index: 20
Arthur Christopoulos
H-Index: 62
Ligand-directed biased agonism at human histamine H3 receptor isoforms across Gαi/o-and β-arrestin2-mediated pathways
Biochemical Pharmacology
2023/12/28
Arthur Christopoulos
H-Index: 62
Design, synthesis and evaluation of novel 2-phenyl-3-(1H-pyrazol-4-yl) pyridine positive allosteric modulators for the M4 mAChR
European Journal of Medicinal Chemistry
2023/10/5
Emma T Van Der Westhuizen
H-Index: 14
Yao Lu
H-Index: 4
Arthur Christopoulos
H-Index: 62
Celine Valant
H-Index: 20
The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors
British journal of pharmacology
2023/10
Arthur Christopoulos
H-Index: 62
George Abraham
H-Index: 3
Geoffrey Burnstock
H-Index: 68
Stefania Ceruti
H-Index: 24
Nan Chiang
H-Index: 47
Olivier Civelli
H-Index: 40
Steven D Douglas
H-Index: 6
Michael L Garelja
H-Index: 6
Karen J Gregory
H-Index: 30
Debbie L Hay
H-Index: 33
Deron Herr
H-Index: 24
Ahsan Husain
H-Index: 24
Pawel Kozielewicz
H-Index: 8
Dan Larhammar
H-Index: 25
Katie Leach
H-Index: 19
Davide Lecca
H-Index: 20
John D Lee
H-Index: 46
Martin C Michel
H-Index: 40
Duuamene Nyimanu
H-Index: 5
Rithwik Ramachandran
H-Index: 22
Gunnar Schulte
H-Index: 31
Stefan Schulz
H-Index: 4
Roger Summers
H-Index: 32
David Thal
H-Index: 14
Xanomeline displays concomitant orthosteric and allosteric binding modes at the M4 mAChR
Nature communications
2023/9/6
Structure-based virtual screening discovers potent and selective adenosine A1 receptor antagonists
European Journal of Medicinal Chemistry
2023/9/5
Jo-Anne Baltos
H-Index: 12
Arthur Christopoulos
H-Index: 62
Jan Kihlberg
H-Index: 26
Lauren Therese May
H-Index: 27
Jens Carlsson
H-Index: 21
Role of conserved tyrosine lid residues in the activation of the M2 muscarinic acetylcholine receptor
Molecular Pharmacology
2023/9/1
Structural basis of efficacy-driven ligand selectivity at GPCRs
Nature Chemical Biology
2023/7
Pharmacological hallmarks of allostery at the M4 muscarinic receptor elucidated through structure and dynamics
Elife
2023/5/30
Acetylcholine receptors (muscarinic) in GtoPdb v. 2023.1
IUPHAR/BPS Guide to Pharmacology CITE
2023/4/26
David A Brown
H-Index: 12
Arthur Christopoulos
H-Index: 62
Chris Langmead
H-Index: 20
David Thal
H-Index: 14
Celine Valant
H-Index: 20
The role of the adenosine system in epilepsy and its comorbidities
2023/4/19
Structural and Molecular Determinants for Isoform Bias at Human Histamine H3 Receptor Isoforms
ACS Chemical Neuroscience
2023/1/26
Arthur Christopoulos
H-Index: 62
Importance of receptor expression in the classification of novel ligands at the M2 muscarinic acetylcholine receptor
British Journal of Pharmacology
2023/1/20
Structure–activity relationship of pyrazol-4-yl-pyridine derivatives and identification of a radiofluorinated probe for imaging the muscarinic acetylcholine receptor M4
Acta Pharmaceutica Sinica B
2023/1/1
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ-Opioid Receptor
Journal of Medicinal Chemistry
2022/9/13
Examining the Role of the Linker in Bitopic N6-Substituted Adenosine Derivatives Acting as Biased Adenosine A1 Receptor Agonists
Journal of Medicinal Chemistry
2022/6/22
Arthur Christopoulos
H-Index: 62
Identification and Preclinical Development of a Radiofluorinated Probe for Imaging the Muscarinic Acetylcholine Receptor M4 by Positron Emission Tomography
2022/6/1
Secretin amino-terminal structure-activity relationships and complementary mutagenesis at the site of docking to the secretin receptor
Molecular pharmacology
2022/6/1
Investigating Drivers for M1 Muscarinic Acetylcholine Receptor‐Mediated Adverse Events by M1 Positive Allosteric Modulators
The FASEB Journal
2022/5
