Peter Scammells
Monash University
H-index: 54
Oceania-Australia
Top articles of Peter Scammells
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Chemoproteomics validates selective targeting of Plasmodium M1 alanyl aminopeptidase as an antimalarial strategy | Darren Creek Carlo Giannangelo Matthew Challis Ghizal Siddiqui Rebecca Edgar | 2023/8/17 | |
Design, synthesis and evaluation of novel 2-phenyl-3-(1H-pyrazol-4-yl) pyridine positive allosteric modulators for the M4 mAChR | European Journal of Medicinal Chemistry | Manuela Jörg Emma T van der Westhuizen Yao Lu KH Christopher Choy David M Shackleford | 2023/10/5 |
Structure-based development of potent Plasmodium falciparum M1 and M17 aminopeptidase selective and dual inhibitors via S1′-region optimisation | European Journal of Medicinal Chemistry | Petar PS Calic Natalie B Vinh Chaille T Webb Tess R Malcolm Anna Ngo | 2023/2/15 |
On-target, dual aminopeptidase inhibition provides cross-species antimalarial activity. | bioRxiv | Rebecca CS Edgar Ghizal Siddiqui Tess R Malcolm Sandra Duffy Mrittika Chowdhury | 2023 |
Biocompatible cationic lipoamino acids as counterions for oral administration of API-ionic liquids | Pharmaceutical Research | Anthony Lai Nathania Leong Dan Zheng Leigh Ford Tri-Hung Nguyen | 2022/10 |
Genetic and chemical validation of Plasmodium falciparum aminopeptidase PfA-M17 as a drug target in the hemoglobin digestion pathway | Elife | Rebecca CS Edgar Ghizal Siddiqui Katheryn Hjerrild Tess R Malcolm Natalie B Vinh | 2022/9/13 |
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ-Opioid Receptor | Journal of Medicinal Chemistry | Owindeep Deo Sadia Alvi Vi Pham Arthur Christopoulos David M Thal | 2022/9/13 |
Examining the Role of the Linker in Bitopic N6-Substituted Adenosine Derivatives Acting as Biased Adenosine A1 Receptor Agonists | Journal of Medicinal Chemistry | Jon Kyle Awalt Anh TN Nguyen Tim J Fyfe Bui San Thai Paul J White | 2022/6/22 |
MAPK inhibitors | 2022/3/15 | ||
Structural features of iperoxo–BQCA muscarinic acetylcholine receptor hybrid ligands determining subtype selectivity and efficacy | ACS Chemical Neuroscience | Matthew CL Wakeham Briana J Davie David K Chalmers Arthur Christopoulos Ben Capuano | 2021/12/14 |
Lipophilic salts and lipid-based formulations: Enhancing the oral delivery of octreotide | Pharmaceutical Research | Peng Li Leigh Ford Shadabul Haque Mitchell P McInerney Hywel D Williams | 2021/6 |
Discovery and development of 2-aminobenzimidazoles as potent antimalarials | European Journal of Medicinal Chemistry | Shane M Devine Matthew P Challis Jomo K Kigotho Ghizal Siddiqui Amanda De Paoli | 2021/10/5 |
Development and Application of Subtype-Selective Fluorescent Antagonists for the Study of the Human Adenosine A1 Receptor in Living Cells | Journal of Medicinal Chemistry | Eleonora Comeo Phuc Trinh Anh T Nguyen Cameron J Nowell Nicholas D Kindon | 2021/3/16 |
Positive allosteric mechanisms of adenosine A1 receptor-mediated analgesia | Nature | Christopher J Draper-Joyce Rebecca Bhola Jinan Wang Apurba Bhattarai Anh TN Nguyen | 2021/9/23 |
Stabilising disproportionation of lipophilic ionic liquid salts in lipid-based formulations | International Journal of Pharmaceutics | Anthony Lai Yasemin Sahbaz Leigh Ford Tri-Hung Nguyen Shadabul Haque | 2021/3/15 |
1, 3‐Benzodioxole‐Modified Noscapine Analogues: Synthesis, Antiproliferative Activity, and Tubulin‐Bound Structure | ChemMedChem | Cassandra Yong Shane M Devine Anne‐Catherine Abel Stefan D Tomlins Divya Muthiah | 2021/9/16 |
A Structure− Activity Relationship Study of Novel Hydroxamic Acid Inhibitors around the S1 Subsite of Human Aminopeptidase N | ChemMedChem | Jisook Lee Nyssa Drinkwater Sheena McGowan Peter Scammells | 2021/1/8 |
Fragment-based development of bacterial DsbA inhibitors as novel anti-virulence agents | Acta Crystallographica Section A: Foundations and Advances | Geqing Wang Wesam Alwan Matthew Bentley Biswaranjan Mohanty Bradley Doak | 2021/8/1 |
Development of Novel 4‐Arylpyridin‐2‐one and 6‐Arylpyrimidin‐4‐one Positive Allosteric Modulators of the M1 Muscarinic Acetylcholine Receptor | ChemMedChem | Manuela Jörg Elham Khajehali Emma T van der Westhuizen KH C. Choy David M Shackleford | 2021/1/8 |
Enantioenriched Positive Allosteric Modulators Display Distinct Pharmacology at the Dopamine D1 Receptor | Molecules | Tim J Fyfe Peter J Scammells J Robert Lane Ben Capuano | 2021/6/22 |
Co-Authors
