Stefan Knapp
Goethe-Universität Frankfurt am Main
H-index: 110
Europe-Germany
Top articles of Stefan Knapp
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Structure-Guided Design of a Highly Potent Partial RXR Agonist with Superior Physicochemical Properties | Journal of Medicinal Chemistry | Max Lewandowski Melania Carmina Loris Knümann Minh Sai Sabine Willems | 2024/1/18 |
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine‐Independent and Chronic Itch | Advanced Science | Annika Balzulat W Felix Zhu Cathrin Flauaus Victor Hernandez‐Olmos Jan Heering | 2024/2/13 |
Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator | Journal of Medicinal Chemistry | Lara Dötsch Caitlin Davies Elisabeth Hennes Julia Schönfeld Adarsh Kumar | 2024/3/12 |
Luciferase-and HaloTag-based reporter assays to measure small-molecule-induced degradation pathway in living cells | Martin P Schwalm Krishna Saxena Susanne Müller Stefan Knapp | 2024/4/18 | |
High throughput screening for LC3/GABARAP binders utilizing fluorescence polarization assay | arXiv preprint arXiv:2401.04453 | Martin P Schwalm Johannes Dopfer Stefan Knapp Vladimir V Rogov | 2024/1/9 |
Inhibition of Parkinson’s disease-related LRRK2 by type-I and type-II kinase inhibitors: Activity and structures | Biophysical Journal | Marta M Sanz Murillo Amalia C Villagran Suarez Verena Dederer Deep Chatterjee Jaime M Alegrio Louro | 2024/2/8 |
The catalytic domain of free or ligand bound histone deacetylase 4 occurs in solution predominantly in closed conformation | Protein Science | Markus Schweipert Thomas Nehls Anton Frühauf Cecilé Debarnot Adarsh Kumar | 2024/3 |
Expanding the ligand spaces for E3 ligases for the design of protein degraders | Rahman Shah Zaib Saleem Martin P Schwalm Stefan Knapp | 2024/4/12 | |
Development of Highly Potent and Selective FGFR4 Inhibitors Based on SNAr Electrophiles | Moritz Schwarz Maksym Kurkunov Florian Wittlinger Ramona Rudalska Guiqun Wang | 2024/1/2 | |
Photosensitization enables Pauson-Khand–type reactions with nitrenes | Science | Fang Li W Felix Zhu Claire Empel Oleksandr Datsenko Adarsh Kumar | 2024/2/2 |
Development of Selective Pyrido[2,3-d]pyrimidin-7(8H)-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors | Journal of Medicinal Chemistry | Marcel Rak Amelie Menge Roberta Tesch Lena M Berger Dimitrios-Ilias Balourdas | 2024/2/29 |
Tetrahydropyridine LIMK inhibitors: Structure activity studies and biological characterization | European Journal of Medicinal Chemistry | Anthony Champiré Rayan Berabez Abdennour Braka Aurélie Cosson Justine Corret | 2024/4/9 |
Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity | bioRxiv | Joshua Gerninghaus Rezart Zhubi Andreas Kraemer Marwah Karim Do Hoang Nhu Tran | 2024 |
Inhibition of Parkinson's disease-related LRRK2 by type-I and type-II kinase inhibitors: Activity and structures | Biophysical Journal | Marta M Sanz Murillo Amalia C Villagran Suarez Verena Dederer Deep Chatterjee Jaime M Alegrio Louro | 2024/2 |
Small Scale purification test for expression of human PINK1 in insect cells | Verena Dederer Olawale G Raimi Miratul MK Muqit Stefan Knapp Sebastian Mathea | 2024/2/19 | |
tracerDB: A crowdsourced fluorescent tracer database for target engagement analysis | Martin Schwalm Johannes Dopfer James Vasta Susanne Muller Stefan Knapp | 2024/3/28 | |
Thermodynamic Characterization of LC3/GABARAP Ligands by Isothermal Titration Calorimetry | bioRxiv | Johannes Dopfer Martin P Schwalm Stefan Knapp Vladimir V Rogov | 2024 |
Development of potent dual BET/HDAC inhibitors via pharmacophore merging and structure-guided optimization | ACS Chemical Biology | Nicolas Bauer Dimitrios-Ilias Balourdas Joel R Schneider Xin Zhang Lena M Berger | 2024/1/31 |
Synthesis and biological evaluation of 1H-pyrrolo [3, 2–g] isoquinolines | Bioorganic & medicinal chemistry letters | Kasa Shiva Raju Sandeep AnkiReddy Gowravaram Sabitha Vagolu Siva Krishna Dharmarajan Sriram | 2019/1/15 |
Development of Highly Potent and Selective Covalent FGFR4 Inhibitors Based on SNAr Electrophiles | Journal of Medicinal Chemistry | Moritz Schwarz Maksym Kurkunov Florian Wittlinger Ramona Rudalska Guiqun Wang | 2024/3/25 |
Co-Authors
