Nader S. Abutaleb
Purdue University
H-index: 24
North America-United States
Top articles of Nader S. Abutaleb
Title | Journal | Author(s) | Publication Date |
---|---|---|---|
Novel phenylthiazoles with a tert-butyl moiety: promising antimicrobial activity against multidrug-resistant pathogens with enhanced ADME properties | RSC advances | Mohamed Hagras Abdelrahman A Abuelkhir Nader S Abutaleb Ahmed M Helal Iten M Fawzy | 2024 |
Diiodohydroxyquinoline for the treatment of clostridium difficile infection | 2023/11/7 | ||
Expanding the structure–activity relationships of alkynyl diphenylurea scaffold as promising antibacterial agents | RSC Medicinal Chemistry | Hanzada T Nour El-Din Mohamed M Elsebaie Nader S Abutaleb Ahmed M Kotb Ahmed S Attia | 2023 |
Evaluation of 1, 3, 4-thiadiazole carbonic anhydrase inhibitors for gut decolonization of vancomycin-resistant enterococci | ACS Medicinal Chemistry Letters | Nader S Abutaleb Annadka Shrinidhi Aloka B Bandara Mohamed N Seleem Daniel P Flaherty | 2023/3/21 |
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates | Journal of Enzyme Inhibition and Medicinal Chemistry | Simone Giovannuzzi Anil Kumar Marapaka Nader S Abutaleb Fabrizio Carta Hsin-Wen Liang | 2023/12/31 |
Arylpyrazole as selective anti‐enterococci; synthesis and biological evaluation of novel derivatives for their antimicrobial efficacy | Journal of Heterocyclic Chemistry | Ahmed M Sayed Nader S Abutaleb Ahmed Kotb Hany G Ezzat Mohamed N Seleem | 2023/1 |
SAR investigation and optimization of benzimidazole-based derivatives as antimicrobial agents against Gram-negative bacteria | European Journal of Medicinal Chemistry | Eman ME Dokla Nader S Abutaleb Sandra N Milik Ezzat AEA Kandil Omar M Qassem | 2023/2/5 |
Discovery of 1, 2-diaryl-3-oxopyrazolidin-4-carboxamides as a new class of MurA enzyme inhibitors and characterization of their antibacterial activity | European Journal of Medicinal Chemistry | Reem A Wagdy Nader S Abutaleb Reem K Fathalla Yehia Elgammal Stefanie Weck | 2023/12/5 |
Colonization efficiency of multidrug-resistant Neisseria gonorrhoeae in a female mouse model | Pathogens and Disease | Babatomiwa Kikiowo Aloka B Bandara Nader S Abutaleb Mohamed N Seleem | 2023 |
Identification of N-(5-nitrothiazol-2-yl)-3-oxopyrazolidine-4-carboxamide derivative as a potent inhibitor of Clostridioides difficile | Reem Wagdy Nader Abutaleb Yehia El-Gammal Rusha Pal Ashraf Abadi | 2023/11/29 | |
Naphthylthiazoles: a class of broad-spectrum antifungals | RSC Medicinal Chemistry | Mohamed Hagras Nader S Abutaleb Hany G Ezzat Ehab A Salama Mohamed N Seleem | 2023 |
Substituted salicylic acid analogs offer improved potency against multidrug-resistant Neisseria gonorrhoeae and good selectivity against commensal vaginal bacteria | Scientific Reports | Hanan Almolhim Ahmed EM Elhassanny Nader S Abutaleb Abdallah S Abdelsattar Mohamed N Seleem | 2023/9/2 |
Exploring novel aryl/heteroaryl-isosteres of phenylthiazole against multidrug-resistant bacteria | RSC advances | Mariam Omara Mohamed Hagras Mohamed M Elsebaie Nader S Abutaleb Hanzada T Nour El-Din | 2023 |
Lopinavir and ritonavir act synergistically with azoles against Candida auris in vitro and in a mouse model of disseminated candidiasis | International Journal of Antimicrobial Agents | Ehab A Salama Hassan E Eldesouky Yehia Elgammal Nader S Abutaleb Mohamed N Seleem | 2023/9/1 |
Isoquinoline antimicrobial agent: Activity against intracellular bacteria and effect on global bacterial proteome | Molecules | Caroline W Karanja Nimishetti Naganna Nader S Abutaleb Neetu Dayal Kenneth I Onyedibe | 2022/8/10 |
Mechanistic Studies and In Vivo Efficacy of an Oxadiazole-Containing Antibiotic | Journal of medicinal chemistry | George A Naclerio Nader S Abutaleb Kenneth I Onyedibe Caroline Karanja Hassan E Eldesouky | 2022/4/28 |
Auranofin exerts antibacterial activity against Neisseria gonorrhoeae in a female mouse model of genital tract infection | PloS one | Ahmed EM Elhassanny Nader S Abutaleb Mohamed N Seleem | 2022/4/21 |
Structure-activity relationship studies for inhibitors for vancomycin-resistant Enterococcus and human carbonic anhydrases | The FASEB Journal | Monica Soto Velasquez Neha Rana Doungkamol Alongkronrusmee Karin FK Ejendal Kwaku Kyei‐Baffour | 2017/4 |
Exploring the structure-activity relationships of diphenylurea as an antibacterial scaffold active against methicillin-and vancomycin-resistant Staphylococcus aureus | European Journal of Medicinal Chemistry | Mohamed M Elsebaie Hanzada T Nour El-Din Nader S Abutaleb Abdelrahman A Abuelkhir Hsin-Wen Liang | 2022/4/15 |
Repurposing FDA-approved sulphonamide carbonic anhydrase inhibitors for treatment of Neisseria gonorrhoeae | Journal of Enzyme Inhibition and Medicinal Chemistry | Nader S Abutaleb Ahmed EM Elhassanny Alessio Nocentini Chad S Hewitt Ahmed Elkashif | 2022/12/31 |