George G. Holz
SUNY Upstate Medical University
H-index: 50
North America-United States
Top articles of George G. Holz
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Corrination Mitigates Peptide Aggregation as Exemplified for Glucagon | Peptides | Amber Liles Nancy Cham Morgan L Opp Ian C Tinsley Oleg G Chepurny | 2024/1/1 |
Excess pancreatic elastase alters acinar-β cell communication by impairing the mechano-signaling and the PAR2 pathways | Cell metabolism | Giorgio Basile Amedeo Vetere Jiang Hu Oluwaseun Ijaduola Yi Zhang | 2023/7/11 |
A peptide triple agonist of GLP-1, neuropeptide Y1, and neuropeptide Y2 receptors promotes glycemic control and weight loss | Scientific reports | Kylie S Chichura Clinton T Elfers Therese S Salameh Varun Kamat Oleg G Chepurny | 2023/6/12 |
GTS-21, a selective alpha7 nicotinic acetylcholine receptor agonist, ameliorates diabetic nephropathy in Leprdb/db mice | Scientific Reports | Qinghe Meng Xinghan Tian Junwei Li Napat Pruekprasert Ravi Dhawan | 2022/12/26 |
Nonpeptidic Z360-Analogs Tagged with Trivalent Radiometals as Anti-CCK2R Cancer Theranostic Agents: A Preclinical Study | Pharmaceutics | Berthold A Nock Panagiotis Kanellopoulos Oleg G Chepurny Maritina Rouchota George Loudos | 2022/3/18 |
The α7nAChR agonist GTS-21 engages the GLP-1 incretin hormone axis to lower levels of blood glucose in db/db mice. | Diabetes, Obesity & Metabolism | Q Meng OG Chepurny CA Leech N Pruekprasert ME Molnar | 2022/3/16 |
Intra-islet glucagon confers β-cell glucose competence for first-phase insulin secretion and favors GLP-1R stimulation by exogenous glucagon | Journal Of Biological Chemistry | Over Cabrera James Ficorilli Janice Shaw Felipe Echeverri Frank Schwede | 2022/2/1 |
Synthesis, in vitro biological investigation, and molecular dynamics simulations of thiazolopyrimidine based compounds as corticotrophin releasing factor receptor-1 antagonists | Bioorganic chemistry | Hossam R Elgiushy Nageh A Abou-Taleb George G Holz Oleg G Chepurny Ioannis Pirmettis | 2021/9/1 |
Cyclic AMP‐dependent activation of ERK via GLP‐1 receptor signalling requires the neuroendocrine cell‐specific guanine nucleotide exchanger NCS‐RapGEF2 | Journal of neuroendocrinology | Wenqin Xu Sam P Dahlke Andrew C Emery Michelle Sung Oleg G Chepurny | 2021/7 |
Synthesis, Optimization, and Biological Evaluation of Corrinated Conjugates of the GLP-1R Agonist Exendin-4 | Journal of Medicinal Chemistry | Ian C Tinsley Tito Borner MacKenzie L Swanson Oleg G Chepurny Sarah A Doebley | 2021/3/6 |
Design and Evaluation of Peptide Dual-Agonists of GLP-1 and NPY2 Receptors for Glucoregulation and Weight Loss with Mitigated Nausea and Emesis | Journal of medicinal chemistry | Brandon T Milliken Clinton Elfers Oleg G Chepurny Kylie S Chichura Ian R Sweet | 2021/1/15 |
Discovery of a stable tripeptide targeting the N-domain of CRF1 receptor | Amino acids | George Liapakis Vlasios Karageorgos Ioannis Andreadelis George G Holz Eirini Dermitzaki | 2020/9 |
[99mTc]Tc-DGA1, a Promising CCK2R-Antagonist-Based Tracer for Tumor Diagnosis with Single-Photon Emission Computed Tomography | Molecular pharmaceutics | Aikaterini Kaloudi Panagiotis Kanellopoulos Thorsten Radolf Oleg G Chepurny Maritina Rouchota | 2020/6/22 |
Corrination of a GLP-1 receptor agonist for glycemic control without emesis | Cell reports | Tito Borner Jayme L Workinger Ian C Tinsley Samantha M Fortin Lauren M Stein | 2020/6/16 |
FRET Reporter Assays for cAMP and Calcium in a 96-well Format Using Genetically Encoded Biosensors Expressed in Living Cells | Bio-Protocol | BT Milliken RP Doyle GG Holz O. Chepurny | 2020/6 |
Therapeutic potential of α7 nicotinic acetylcholine receptor agonists to combat obesity, diabetes, and inflammation | Han Xie Natesh Yepuri Qinghe Meng Ravi Dhawan Colin A Leech | 2020/12 |
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