Xerardo García Mera, ORCID 0000-0001-5218-6351
Universidad de Santiago de Compostela
H-index: 28
Europe-Spain
Top articles of Xerardo García Mera, ORCID 0000-0001-5218-6351
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Exploring structural determinants of neuroprotection bias on novel glypromate conjugates with bioactive amines | European Journal of Medicinal Chemistry | Sara C Silva-Reis Vera M Costa Daniela Correia da Silva David M Pereira Xavier Cruz Correia | 2024/3/5 |
Exploring Biginelli-based scaffolds as A2B adenosine receptor antagonists: Unveiling novel structure-activity relationship trends, lead compounds, and potent colorectal … | Biomedicine & pharmacotherapy | Rubén Prieto-Díaz Hugo Fojo-Carballo Maria Majellaro Tana Tandarić Jhonny Azuaje | 2024/4/1 |
Concise overview of glypromate neuropeptide research: from chemistry to pharmacological applications in neurosciences | Sara C Silva-Reis Ivo E Sampaio-Dias Vera M Costa Xavier Cruz Correia Hugo F Costa-Almeida | 2023/2/3 | |
Pharmacological insights emerging from the characterization of a large collection of synthetic cannabinoid receptor agonists designer drugs | Biomedicine & Pharmacotherapy | Claudia Gioé-Gallo Sandra Ortigueira José Brea Iu Raïch Jhonny Azuaje | 2023/8/1 |
P27. Discovery of glypromate conjugates with biomedical applications in Alzheimer’s disease | Book of Abstracts | Sara C Silva-Reis Ivo E Sampaio-Dias Daniela Correia da Silva Xavier C Correia Hugo F Costa-Almeida | 2023/2/10 |
Stapling Amantadine to Melanostatin Neuropeptide: Discovery of Potent Positive Allosteric Modulators of the D2 Receptors | ACS Medicinal Chemistry Letters | Sara C Silva-Reis Xavier C Correia Hugo F Costa-Almeida Beatriz L Pires-Lima Daiane Maronde | 2023/11/14 |
Exploring Non-orthosteric Interactions with a Series of Potent and Selective A3 Antagonists | ACS Medicinal Chemistry Letters | Darío Miranda-Pastoriza Rodrigo Bernárdez Jhonny Azuaje Rubén Prieto-Díaz Maria Majellaro | 2022/1/10 |
Exploring the Effect of Halogenation in a Series of Potent and Selective A2B Adenosine Receptor Antagonists | Journal of Medicinal Chemistry | Rubén Prieto-Díaz Manuel González-Gómez Hugo Fojo-Carballo Jhonny Azuaje Abdelaziz El Maatougui | 2022/12/14 |
Optimization of 2-Amino-4, 6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1 Antagonists | Cristina Val García Carlos Rodríguez García Rubén Prieto Díaz Abel Crespo Gavilán Jhonny Alberto Azuaje Guerrero | 2022 | |
A2B adenosine receptor antagonists rescue lymphocyte activity in adenosine-producing patient-derived cancer models | Journal for Immunotherapy of Cancer | Apple Hui Min Tay Rubén Prieto-Díaz Shiyong Neo Le Tong Xinsong Chen | 2022 |
A Chemical Strategy to Improve Bioavailability of Glypromate Peptide-Conjugates | Sara C Silva-Reis Ivo E Sampaio-Dias Hugo F Costa-Almeida Vera M Costa Xerardo García-Mera | 2022/11/1 | |
Isolation and structural characterization of stable carbamic–carbonic anhydrides: an experimental and computational study | Organic Chemistry Frontiers | Ivo E Sampaio-Dias Carlos AD Sousa Sara C Silva-Reis Luís Pinto da Sílva Xerardo García-Mera | 2022 |
Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1 Antagonists | Journal of Medicinal Chemistry | Cristina Val Carlos Rodríguez-García Rubén Prieto-Díaz Abel Crespo Jhonny Azuaje | 2022/1/22 |
Catalytic performance of a metal-free graphene oxide-Al2O3 composite assembled by 3D printing | Journal of the European Ceramic Society | Jhonny Azuaje Adrián Rama Ana Mallo-Abreu Mónica G Boado María Majellaro | 2021/2/1 |
Exploring the bioisosterism of proline residue in melanostatin neuropeptide using heteroaromatic scaffolds | Beatriz L Pires-Lima Sara Silva-Reis Xavier Cruz Correia Hugo Costa-Almeida Xerardo García-Mera | 2021/11/3 | |
PTML Computational Study, Synthesis, and Pharmacological Assay of MIF-1 Peptidomimetics | Ivo Sampaio Jose Borges Jose Brea Dolores Viña Mabel Losa | 2021/1/7 | |
Using aza-proline for the assembly of a melanostatin aza-peptide derivative | Xavier Cruz Correia Sara C Silva-Reis Beatriz L Pires-Lima Hugo F Costa-Almeida Xerardo García-Mera | 2021/11/3 | |
Synthesis, Pharmacological, and Biological Evaluation of 2-Furoyl-Based MIF-1 Peptidomimetics and the Development of a General-Purpose Model for Allosteric Modulators (ALLOPTML) | ACS Chemical Neuroscience | Ivo E Sampaio-Dias José E Rodríguez-Borges Víctor Yáñez-Pérez Sonia Arrasate Javier Llorente | 2021 |
Design, synthesis, and biological evaluation of hybrid glypromate analogues using 2-azanorbornane as a prolyl and pipecolyl surrogate | ACS Chemical Neuroscience | Ivo E Sampaio-Dias Miguel Santejo Sara C Silva-Reis Marcia A Liz Cristina Alcoholado | 2021/9/13 |
Potent and Subtype-Selective Dopamine D2 Receptor Biased Partial Agonists Discovered via an Ugi-Based Approach | Journal of Medicinal Chemistry | Ana Mallo-Abreu Irene Reyes-Resina Jhonny Azuaje Rafael Franco Aitor García-Rey | 2021/6/10 |
Co-Authors
