Oriana Tabarrini
Università degli Studi di Perugia
H-index: 38
Europe-Italy
Top articles of Oriana Tabarrini
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Synthetically accessible de novo design using reaction vectors: Application to PARP1 inhibitors | Molecular Informatics | Gian Marco Ghiandoni Stuart R Flanagan Michael J Bodkin Maria Giulia Nizi Albert Galera‐Prat | 2024/2/6 |
Switching the three-component Biginelli-like reaction conditions for the regioselective synthesis of new 2-amino [1, 2, 4] triazolo [1, 5-a] pyrimidines | Organic & Biomolecular Chemistry | Martina Pacetti Maria Chiara Pismataro Tommaso Felicetti Federica Giammarino Anna Bonomini | 2024 |
Privileged scaffolds for potent and specific inhibitors of mono-ADP-ribosylating PARPs | Maria Giulia Nizi Chiara Sarnari Oriana Tabarrini | 2023/8/3 | |
[1,2,4]Triazolo[3,4-b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes | Journal of Medicinal Chemistry | Sudarshan Murthy Maria Giulia Nizi Mirko M Maksimainen Serena Massari Juho Alaviuhkola | 2023/1/4 |
Compounds for use in the treatment of cancer and inflammatory conditions | L Lehtiö M Maksimainen N Murthy Sudarshan O Tabarrini MG Nizi | 2023 | |
From Serendipity to Rational Identification of the 5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4(3H)-one Core as a New Chemotype of AKT1 Inhibitors for … | Pharmaceutics | Andrea Astolfi Francesca Milano Deborah Palazzotti Jose Brea Maria Chiara Pismataro | 2022/10/26 |
Potent 2, 3-dihydrophthalazine-1, 4-dione derivatives as dual inhibitors for mono-ADP-ribosyltransferases PARP10 and PARP15 | European Journal of Medicinal Chemistry | Maria Giulia Nizi Mirko M Maksimainen Sudarshan Murthy Serena Massari Juho Alaviuhkola | 2022/7/5 |
Medicinal chemistry perspective on targeting mono-ADP-ribosylating PARPs with small molecules | Maria Giulia Nizi Mirko M Maksimainen Lari Lehtio Oriana Tabarrini | 2022/5/24 | |
Discovery of 2-phenylquinolines with broad-spectrum anti-coronavirus activity | ACS Medicinal Chemistry Letters | Maria Giulia Nizi Leentje Persoons Angela Corona Tommaso Felicetti Giada Cernicchi | 2022/5/3 |
Triazolopyrimidine Nuclei: Privileged Scaffolds for Developing Antiviral Agents with a Proper Pharmacokinetic Profile | Tommaso Felicetti Maria C Pismataro Violetta Cecchetti Oriana Tabarrini Serena Massari | 2022/3/1 | |
New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains | European Journal of Medicinal Chemistry | Tommaso Felicetti Nicholas Cedraro Andrea Astolfi Giada Cernicchi Gianmarco Mangiaterra | 2022/11/5 |
From Quinoline to Quinazoline‐Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search | ChemMedChem | Nicholas Cedraro Rolando Cannalire Andrea Astolfi Gianmarco Mangiaterra Tommaso Felicetti | 2021/10/6 |
1, 2, 4-Triazolo [1, 5-a] pyrimidines: Efficient one-step synthesis and functionalization as influenza polymerase PA-PB1 interaction disruptors | European Journal of Medicinal Chemistry | Maria Chiara Pismataro Tommaso Felicetti Chiara Bertagnin Maria Giulia Nizi Anna Bonomini | 2021/10/5 |
Sustainable, three-component, one-pot procedure to obtain active anti-flavivirus agents | European Journal of Medicinal Chemistry | Tommaso Felicetti Maria Sole Burali Chin Piaw Gwee Kitti Wing Ki Chan Sylvie Alonso | 2021/1/15 |
Synthesis and characterization of 1, 2, 4-triazolo [1, 5-a] pyrimidine-2-carboxamide-based compounds targeting the PA-PB1 interface of influenza A virus polymerase | European journal of medicinal chemistry | Serena Massari Chiara Bertagnin Maria Chiara Pismataro Anna Donnadio Giulio Nannetti | 2021/1/1 |
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors | Journal of Enzyme Inhibition and Medicinal Chemistry | Tommaso Felicetti Gianmarco Mangiaterra Rolando Cannalire Nicholas Cedraro Donatella Pietrella | 2020/1/1 |
Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors | International Journal of Molecular Sciences | Rolando Cannalire Gianmarco Mangiaterra Tommaso Felicetti Andrea Astolfi Nicholas Cedraro | 2020/9/24 |
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors | European Journal of Medicinal Chemistry | Maria Giulia Nizi Jenny Desantis Yoshio Nakatani Serena Massari Maria Angela Mazzarella | 2020/9/1 |
Corso di Laurea Magistrale in Chimica e Tecnologia Farmaceutiche | Oriana Presidente TABARRINI Stefano GIOVAGNOLI Francesca FALLARINO Luana PERIOLI Andrea TEMPERINI | 2020/5/9 | |
Pyridobenzothiazolones exert potent anti-dengue activity by hampering multiple functions of NS5 polymerase | ACS Medicinal Chemistry Letters | Rolando Cannalire Kitti Wing Ki Chan Maria Sole Burali Chin Piaw Gwee Sai Wang | 2020/3/19 |
