Ondřej Benek
Univerzita Hradec Králové
H-index: 15
Europe-Czech Republic
Top articles of Ondřej Benek
Title | Journal | Author(s) | Publication Date |
---|---|---|---|
Nanomolar Benzothiazole-Based Inhibitors of 17β-HSD10 with Cellular Bioactivity | ACS Medicinal Chemistry Letters | Michaela Hanzlova Marketa Sedlacek Miskerikova Aneta Rotterova Katarina Chalupova Katarina Jurkova | 2023/11/10 |
Development of Submicromolar 17β-HSD10 inhibitors and their in vitro and in vivo evaluation | European Journal of Medicinal Chemistry | Ondrej Benek Michaela Vaskova Marketa Miskerikova Monika Schmidt Rudolf Andrys | 2023/10/5 |
Physiologically relevant fluorescent assay for identification of 17β‐hydroxysteroid dehydrogenase type 10 inhibitors | Journal of Neurochemistry | Monika Schmidt Michaela Vaskova Aneta Rotterova Pavlina Fiandova Marketa Miskerikova | 2023/10 |
Small‐molecule inhibitors of cyclophilin D as potential therapeutics in mitochondria‐related diseases | Annamaria Haleckova Ondrej Benek Lucie Zemanová Rafael Dolezal Kamil Musilek | 2022/9 | |
Effects of novel 17β-hydroxysteroid dehydrogenase type 10 inhibitors on mitochondrial respiration | Toxicology Letters | Zdeněk Fišar Kamil Musílek Ondřej Benek Lukáš Hroch Lucie Vinklářová | 2021/3/15 |
RNase T1 Refolding Assay for Determining Mitochondrial Cyclophilin D Activity: A Novel In Vitro Method Applicable in Drug Research and Discovery | Biochemistry | Lucie Zemanova Michaela Vaskova Monika Schmidt Jana Roubalova Annamaria Haleckova | 2020/4/10 |
SEARCHING FOR NEW ANTIMICROBIAL AGENTS BY TARGETING BACTERIAL NAD METABOLISM: EVALUATION OF FRENTIZOLE DERIVATIVES SELECTED BY MOLECULAR DOCKING. | Military Medical Science Letters/Vojenské Zdravotnické Listy | Michaela Hympanova Tomas Kucera Ondrej Benek Jan Korabecny Jan Marek | 2020/4/1 |
Friend or enemy? Review of 17β‐HSD10 and its role in human health or disease | Lucie Vinklarova Monika Schmidt Ondrej Benek Kamil Kuca Frank Gunn‐Moore | 2020/11 | |
Benzothiazolyl ureas are low micromolar and uncompetitive inhibitors of 17β-HSD10 with implications to Alzheimer’s disease treatment | International Journal of Molecular Sciences | Monika Schmidt Ondrej Benek Lucie Vinklarova Martina Hrabinova Lucie Zemanova | 2020/3/17 |
Exploring the chemical space of benzothiazole-based DNA gyrase B inhibitors | ACS medicinal chemistry letters | Žiga Skok Michaela Barančoková Ondřej Benek Cristina Durante Cruz Päivi Tammela | 2020/10/15 |
Discovery of novel berberine derivatives with balanced cholinesterase and prolyl oligopeptidase inhibition profile | European journal of medicinal chemistry | Katerina Sobolova Martina Hrabinova Vendula Hepnarova Tomas Kucera Tereza Kobrlova | 2020/10/1 |
A perspective on multi-target drugs for Alzheimer’s disease | Ondrej Benek Jan Korabecny Ondrej Soukup | 2020/7/1 |