MARGHERITA Brindisi

About MARGHERITA Brindisi

MARGHERITA Brindisi, With an exceptional h-index of 36 and a recent h-index of 29 (since 2020), a distinguished researcher at Università degli Studi di Napoli Federico II, specializes in the field of Medicinal Chemistry-Drug Design-Organic Chemistry.

His recent articles reflect a diverse array of research interests and contributions to the field:

Enantioselective catalytic Strecker reaction on cyclic (Z)-aldimines in flow: reaction optimization and sustainability aspects

Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds

Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray …

Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds

Mechanochemical Fischer indolisation: an eco-friendly design for a timeless reaction

Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route

Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis

Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution

MARGHERITA Brindisi Information

University

Position

- Purdue University

Citations(all)

4660

Citations(since 2020)

3148

Cited By

2740

hIndex(all)

36

hIndex(since 2020)

29

i10Index(all)

84

i10Index(since 2020)

69

Email

University Profile Page

Università degli Studi di Napoli Federico II

Google Scholar

View Google Scholar Profile

MARGHERITA Brindisi Skills & Research Interests

Medicinal Chemistry-Drug Design-Organic Chemistry

Top articles of MARGHERITA Brindisi

Title

Journal

Author(s)

Publication Date

Enantioselective catalytic Strecker reaction on cyclic (Z)-aldimines in flow: reaction optimization and sustainability aspects

Journal of Flow Chemistry

Antonella Ilenia Alfano

Andrea Sorato

Alessia Ciogli

Heiko Lange

Margherita Brindisi

2023/7/19

Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds

ACS Medicinal Chemistry Letters

Antonella Ilenia Alfano

Sveva Pelliccia

Giacomo Rossino

Orazio Chianese

Vincenzo Summa

...

2023/4/12

Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray …

European Journal of Medicinal Chemistry

Irina Stefanelli

Angela Corona

Carmen Cerchia

Emilia Cassese

Salvatore Improta

...

2023/5/5

Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds

ACS Medicinal Chemistry Letters

Antonella Ilenia Alfano

Sveva Pelliccia

Giacomo Rossino

Orazio Chianese

Vincenzo Summa

...

2023/2/3

Mechanochemical Fischer indolisation: an eco-friendly design for a timeless reaction

Green Chemistry

Andrea Porcheddu

Rita Mocci

Margherita Brindisi

Federico Cuccu

Claudia Fattuoni

...

2022

Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route

European Journal of Medicinal Chemistry

Sveva Pelliccia

Carmen Cerchia

Francesca Esposito

Rolando Cannalire

Angela Corona

...

2022/12/15

Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis

European Journal of Pharmacology

Margherita Brindisi

Simona Barone

Alice Rossi

Emilia Cassese

Nunzio Del Gaudio

...

2022/12/5

Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution

Antonella Ilenia Alfano

Heiko Lange

Margherita Brindisi

2022/3/22

Exploring the structural determinants for inhibitor selectivity towards the BACE protein family using structure-based molecular design

Biophysical Journal

Emma K Lendy

Yu-Chen Yen

Emilio L Cardenas

Margherita Brindisi

Arun K Ghosh

...

2022/2/11

Chasing a Breath of Fresh Air in Cystic Fibrosis (CF): Therapeutic Potential of Selective HDAC6 Inhibitors to Tackle Multiple Pathways in CF Pathophysiology

Simona Barone

Emilia Cassese

Antonella Ilenia Alfano

Margherita Brindisi

Vincenzo Summa

2022/2/11

Coupling Interrupted Fischer and Multicomponent Joullié‐Ugi to Chase Chemical Diversity: from Batch to Sustainable Flow Synthesis of Peptidomimetics

ChemMedChem

Antonella Ilenia Alfano

Elisabetta Buommino

Maria Grazia Ferraro

Carlo Irace

Angela Zampella

...

2021/12/14

Harnessing the Role of HDAC6 in Idiopathic Pulmonary Fibrosis: Design, Synthesis, Structural Analysis, and Biological Evaluation of Potent Inhibitors

Journal of medicinal chemistry

Giuseppe Campiani

Caterina Cavella

Jeremy D Osko

Margherita Brindisi

Nicola Relitti

...

2021/7/12

Flow synthesis approaches to privileged scaffolds–recent routes reviewed for green and sustainable aspects

Green Chemistry

Antonella Ilenia Alfano

Margherita Brindisi

Heiko Lange

2021

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–7

Arduino A Mangoni

Jean Jacques Vanden Eynde

Josef Jampilek

Dimitra Hadjipavlou-Litina

Hong Liu

...

2019/6/30

Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological Evaluation

ACS Medicinal Chemistry Letters

A Prasanth Saraswati

Nicola Relitti

Margherita Brindisi

Jeremy D Osko

Giulia Chemi

...

2020/9/29

Drug development and medicinal chemistry efforts toward SARS‐coronavirus and Covid‐19 therapeutics

Arun K Ghosh

Margherita Brindisi

Dana Shahabi

Mackenzie E Chapman

Andrew D Mesecar

2020/6/4

Autophagy modulators for the treatment of oral and esophageal squamous cell carcinomas

Tuhina Khan

Nicola Relitti

Margherita Brindisi

Stefania Magnano

Daniela Zisterer

...

2020/5

Telomerase-based cancer therapeutics: a review on their clinical trials

Nicola Relitti

Akella P Saraswati

Stefano Federico

Tuhina Khan

Margherita Brindisi

...

2020/3/1

Novel quinolone-based potent and selective HDAC6 inhibitors: synthesis, molecular modelling studies and biological investigation

European Journal of Medicinal Chemistry

Nicola Relitti

A Prasanth Saraswati

Giulia Chemi

Margherita Brindisi

Simone Brogi

...

2021/2/15

Harnessing interrupted Fischer in continuous flow: sustainable synthesis of (spiro) indolenine and (spiro) indoline privileged scaffolds

Reaction Chemistry & Engineering

Antonella Ilenia Alfano

Angela Zampella

Ettore Novellino

Margherita Brindisi

Heiko Lange

2020

See List of Professors in MARGHERITA Brindisi University(Università degli Studi di Napoli Federico II)