Laurent Chiarelli
Università degli Studi di Pavia
H-index: 35
Europe-Italy
Top articles of Laurent Chiarelli
Title | Journal | Author(s) | Publication Date |
---|---|---|---|
Structural basis for specific inhibition of salicylate synthase from Mycobacterium abscessus | European Journal of Medicinal Chemistry | Matteo Mori Mario Cocorullo Andrea Tresoldi Giulia Cazzaniga Arianna Gelain | 2024/2/5 |
Benzothiozinone derivatives with anti-tubercular Activity− Further side chain investigation | European Journal of Medicinal Chemistry | Xiaomei Wu Wenxin Wang Giovanni Stelitano Olga Riabova Bin Wang | 2024/1/15 |
Iron acquisition and metabolism as a promising target for antimicrobials (bottlenecks and opportunities): where do we stand? | Giovanni Stelitano Mario Cocorullo Matteo Mori Stefania Villa Fiorella Meneghetti | 2023/3/24 | |
Optimizing the drug discovery process for the development of MbtI inhibitors as promising anti-virulence agents against TB | M Mori G Cazzaniga A Tresoldi A Gelain LR Chiarelli | 2023/9/21 | |
Mycobacterium abscessus Infections in Cystic Fibrosis Individuals: A Review on Therapeutic Options | Deborah Recchia Giovanni Stelitano Alessandro Stamilla Damaris L Gutierrez Giulia Degiacomi | 2023/2/27 | |
Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients? | International Journal of Molecular Sciences | Maura D’Amato Monica Campagnoli Paolo Iadarola Paola Margherita Bignami Marco Fumagalli | 2023/8/31 |
Targeting siderophore-mediated iron uptake in M. abscessus: a new strategy to limit the virulence of non-tuberculous mycobacteria | Pharmaceutics | Matteo Mori Giovanni Stelitano Giulia Cazzaniga Arianna Gelain Andrea Tresoldi | 2023/2 |
Side Chain-Modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity | Biomedicines | Dongguang Fan Bin Wang Giovanni Stelitano Karin Savková Olga Riabova | 2023/7/12 |
Mycobacterium abscessus siderophores biosynthesis as a target to inhibit the iron uptake mechanism | Mario Cocorullo Giovanni Stelitano Matteo Mori Giulia Cazzaniga Martina Roversi | 2023 | |
Improving protection to prevent bacterial infections: preliminary applications of reverse vaccinology against the main cystic fibrosis pathogens | Mario Cocorullo Laurent R Chiarelli Giovanni Stelitano | 2023/7/9 | |
Ironing out Fe3+ acquisition in M. abscessus: a new strategy to target virulence factors in non-tuberculous mycobacteria | M Mori A Tresoldi G Cazzaniga A Gelain G Stelitano | 2023/11/14 | |
From virulence factors to drug development: MbtI as an effective Mycobacterium tuberculosis target | Giovanni Stelitano Mario Cocorullo Giulia Cazzaniga Matteo Mori Stefania Villa | 2023 | |
CanB, a Druggable Cellular Target in Mycobacterium tuberculosis | ACS omega | Giulia Degiacomi Beatrice Gianibbi Deborah Recchia Giovanni Stelitano Giuseppina Ivana Truglio | 2023/7/3 |
Structural Study of a New MbtI-Inhibitor Complex: Towards an Optimized Model for Structure-Based Drug Discovery | Pharmaceuticals | Matteo Mori Stefania Villa Laurent R Chiarelli Fiorella Meneghetti Marco Bellinzoni | 2023/11/3 |
Synthesis, crystal structure, Hirshfeld surface, computational and antibacterial studies of a 9-phenanthrenecarboxaldehyde-based thiodihydropyrimidine derivative | Journal of Molecular Structure | Alakbar Huseynzada Matteo Mori Fiorella Meneghetti Aygun Israyilova Gamze Tuzun | 2022/11/5 |
Crystal Structure, Hirshfeld Surface Analysis, In-Silico and Antimycotic Investigations of Methyl 6-methyl-4-(4-nitrophenyl)-2-oxo-1, 2-dihydropyrimidine-5-carboxylate | Crystals | Alakbar Huseynzada Matteo Mori Fiorella Meneghetti Aygun Israyilova Elif Guney | 2022/12/27 |
WS01. 04 A new weapon against Mycobacterium abscessus | Journal of Cystic Fibrosis | G Degiacomi LR Chiarelli L Muñoz-Muñoz D Recchia G Stelitano | 2022/6/1 |
Phagocyte-targeting polymersomes as intracellular delivery carriers for enzymatic inhibitors with antitubercular activity | G Cazzaniga M Mori F Meneghetti LR Chiarelli G Stelitano | 2022/10/24 | |
A New Benzothiazolthiazolidine Derivative, 11726172, Is Active In Vitro, In Vivo, and against Nonreplicating Cells of Mycobacterium tuberculosis | Msphere | Elena G Salina Umberto Postiglione Laurent R Chiarelli Deborah Recchia Monika Záhorszká | 2022/12/21 |
Virtual screening and crystallographic studies reveal an unexpected γ-lactone derivative active against MptpB as a potential antitubercular agent | European Journal of Medicinal Chemistry | Giulia Cazzaniga Matteo Mori Fiorella Meneghetti Laurent R Chiarelli Giovanni Stelitano | 2022/4/15 |