Koen Augustyns
Universiteit Antwerpen
H-index: 53
Europe-Belgium
Top articles of Koen Augustyns
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Active site-directed probes targeting dipeptidyl peptidases 8 and 9 | European Journal of Medicinal Chemistry | Margarida Espadinha Joni De Loose Sam Corthaut Sofie Thys Yentl Van Rymenant | 2024/4/3 |
A high-throughput target-based screening approach for the identification and assessment of Mycobacterium tuberculosis mycothione reductase inhibitors | Microbiology Spectrum | Natalia Smiejkowska Lauren Oorts Kevin Van Calster Linda De Vooght Rob Geens | 2024/2/5 |
Druglike, ¹⁸F-labeled PET tracers targeting fibroblast activation protein (FAP) | Journal of medicinal chemistry.-Washington, DC, 1963, currens | Muhammet Tanc Nicolò Filippi Yentl Van Rymenant Sergei Grintsevich Isabel Pintelon | 2024 |
Design and Synthesis of 1, 3-Diarylpyrazoles and Investigation of Their Cytotoxicity and Antiparasitic Profile | International Journal of Molecular Sciences | Murat Bozdag Freke Mertens An Matheeussen Natascha Van Pelt Kenn Foubert | 2024/1 |
Druglike, 18F-labeled PET Tracers Targeting Fibroblast Activation Protein | Journal of Medicinal Chemistry | Muhammet Tanc Nicolò Filippi Yentl Van Rymenant Sergei Grintsevich Isabel Pintelon | 2024/4/24 |
Bis (acetamidophenyl) guanidinophenylethylphosphonates for use in the prevention and/or treatment of PAR-related diseases | 2023/5/2 | ||
Beyond ferrostatin-1: a comprehensive review of ferroptosis inhibitors | Camilla Scarpellini Greta Klejborowska Caroline Lanthier Behrouz Hassannia Tom Vanden Berghe | 2023/12/1 | |
From PERK to RIPK1: Design, synthesis and evaluation of novel potent and selective necroptosis inhibitors | Frontiers in Chemistry | Camilla Scarpellini Sophie Valembois Kenneth Goossens Mike Vadi Caroline Lanthier | 2023/4/7 |
Effect of erythrophagocytosis-induced ferroptosis during angiogenesis in atherosclerotic plaques | Angiogenesis | Pauline Puylaert Lynn Roth Melissa Van Praet Isabel Pintelon Catalina Dumitrascu | 2023/11 |
To Target or Not to Target Schistosoma mansoni Cyclic Nucleotide Phosphodiesterase 4A? | International journal of molecular sciences | Yang Zheng Susanne Schroeder Georgi K Kanev Sanaa S Botros Samia William | 2023/4/6 |
Characterization of Structurally Diverse 18F-Labeled d-TCO Derivatives as a PET Probe for Bioorthogonal Pretargeted Imaging | ACS omega | Karuna Adhikari Jonatan Dewulf Christel Vangestel Pieter Van der Veken Sigrid Stroobants | 2023/10/8 |
Chemically diverse activity-based probes with unexpected inhibitory mechanisms targeting trypsin-like serine proteases | Frontiers in Chemistry | Alba Ramos-Llorca Lisse Decraecker Valérie MY Cacheux Irena Zeiburlina Michelle De Bruyn | 2023/1/5 |
Highly Selective Inhibitors of Dipeptidyl Peptidase 9 (DPP9) Derived from the Clinically Used DPP4-Inhibitor Vildagliptin | Journal of Medicinal Chemistry | Siham Benramdane Joni De Loose Nicolò Filippi Margarida Espadinha Olivier Beyens | 2023/9/18 |
The potential role of regulated cell death in dry eye diseases and ocular surface dysfunction | Camilla Scarpellini Alba Ramos Llorca Caroline Lanthier Greta Klejborowska Koen Augustyns | 2023/1/1 | |
Ferroptosis contributes to multiple sclerosis and its pharmacological targeting suppresses experimental disease progression | Cell Death & Differentiation | Emily Van San Angela C Debruyne Geraldine Veeckmans Yulia Y Tyurina Vladimir A Tyurin | 2023/9 |
Selected strategies to fight pathogenic bacteria | Aiva Plotniece Arkadij Sobolev Claudiu T Supuran Fabrizio Carta Fredrik Björkling | 2023/12/31 | |
Targeting ferroptosis protects against experimental (multi) organ dysfunction and death | Nature communications | Samya Van Coillie Emily Van San Ines Goetschalckx Bartosz Wiernicki Banibrata Mukhopadhyay | 2022/2/24 |
A novel ferroptosis inhibitor UAMC-3203, a potential treatment for corneal epithelial wound | Pharmaceutics | Anusha Balla Bao Tran Annika Valtari Philipp Steven Camilla Scarpellini | 2022/12/29 |
Proteases and their potential role as biomarkers and drug targets in dry eye disease and ocular surface dysfunction | Alba Ramos-Llorca Camilla Scarpellini Koen Augustyns | 2022/8/29 | |
Vildagliptin‐Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8/9‐Specific Lead | ChemMedChem | Siham Benramdane Joni De Loose Olivier Beyens Yentl Van Rymenant Gwendolyn Vliegen | 2022/8/3 |
