Jeffrey W Keillor
Ottawa University
H-index: 41
North America-United States
Top articles of Jeffrey W Keillor
Conformational Modulation of Tissue Transglutaminase via Active Site Thiol Alkylating Agents: Size Does Not Matter
Biomolecules
2024/4/19
Jeffrey W Keillor
H-Index: 22
Transcriptomics studies reveal functions of Transglutaminase 2 in breast cancer cells using membrane permeable and impermeable inhibitors
Journal of Molecular Biology
2024/4/10
Fitting of kinact and KI Values from Endpoint Pre-incubation IC50 Data
ACS Medicinal Chemistry Letters
2024/4/4
Jeffrey W Keillor
H-Index: 22
Stabilizing transglutaminase 2 in the open conformation results in reactive astrocytes being more neurosupportive
bioRxiv
2024
Jeffrey W Keillor
H-Index: 22
Metabolic characterisation of transglutaminase 2 inhibitor effects in breast cancer cell lines
The FEBS Journal
2023/11
Elena Ferrari
H-Index: 28
Cristian Taccioli
H-Index: 26
Stefano Volinia
H-Index: 65
Jeffrey W Keillor
H-Index: 22
Nicoletta Bianchi
H-Index: 25
High-Affinity Fluorogenic Substrate for Tissue Transglutaminase Reveals Enzymatic Hysteresis
Biochemistry
2023/10/19
Yasaman Heidari
H-Index: 4
Jeffrey W Keillor
H-Index: 22
Transglutaminase 2 binds to the CD44v6 cytoplasmic domain to stimulate CD44v6/ERK1/2 signaling and maintain an aggressive cancer phenotype
Molecular Cancer Research
2023/9/1
Cell-impermeable inhibitors confirm that intracellular human transglutaminase 2 is responsible for the transglutaminase-associated cancer phenotype
International Journal of Molecular Sciences
2023/8/8
Nicoletta Bianchi
H-Index: 25
Jeffrey W Keillor
H-Index: 22
Targeting transglutaminase 2 mediated exostosin glycosyltransferase 1 signaling in liver cancer stem cells with acyclic retinoid
Cell Death & Disease
2023/6/13
Quinazoline-2-Carboxamides as Selective PET Radiotracers for Matrix Metalloproteinase-13 Imaging in Atherosclerosis
Journal of Medicinal Chemistry
2023/5/9
Jeffrey W Keillor
H-Index: 22
A kinetic study of thiol addition to N-phenylchloroacetamide
Organic & Biomolecular Chemistry
2023
Jeffrey W Keillor
H-Index: 22
A mechanistic study of thiol addition to N-acryloylpiperidine
Organic & Biomolecular Chemistry
2023
Jeffrey W Keillor
H-Index: 22
Peptidic Inhibitors and a Fluorescent Probe for the Selective Inhibition and Labelling of Factor XIIIa Transglutaminase.
Molecules
2023/2/8
Jeffrey W Keillor
H-Index: 22
Novel irreversible peptidic inhibitors of transglutaminase 2
RSC Medicinal Chemistry
2023
The war on hTG2: warhead optimization in small molecule human tissue transglutaminase inhibitors
RSC Medicinal Chemistry
2023
Structure-activity relationships of N-terminal variants of peptidomimetic tissue transglutaminase inhibitors
European Journal of Medicinal Chemistry
2022/3/15
Neda Firoozi
H-Index: 5
Jeffrey W Keillor
H-Index: 22
A mechanistic study of thiol addition to N-phenylacrylamide
Organic & Biomolecular Chemistry
2022
Jeffrey W Keillor
H-Index: 22
Structure–activity relationships of hydrophobic alkyl acrylamides as tissue transglutaminase inhibitors
RSC Medicinal Chemistry
2022
Jeffrey W Keillor
H-Index: 22
Dysregulation of Transglutaminase type 2 through GATA3 defines aggressiveness and Doxorubicin sensitivity in breast cancer
International Journal of Biological Sciences
2022
Cristian Taccioli
H-Index: 26
Jeffrey W Keillor
H-Index: 22
Stefano Volinia
H-Index: 65
Nicoletta Bianchi
H-Index: 25
Sulforaphane covalently interacts with the transglutaminase 2 cancer maintenance protein to alter its structure and suppress its activity
Molecular carcinogenesis
2022/1
Purushottamachar Puranik
H-Index: 12
Jeffrey W Keillor
H-Index: 22
Co-Authors
