James McKerrow
University of California, San Diego
H-index: 107
North America-United States
Top articles of James McKerrow
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
A Single-dose Phase 1 Study With SLV213 Demonstrates Safety and Pharmacokinetics Enabling Investigation of a New Orally Available Cathepsin L Inhibitor for Treatment of … | T Daley K Krantz D Maneval S Simpson J McKerrow | 2024/5 | |
Human schistosomiasis in Nigeria: present status, diagnosis, chemotherapy, and herbal medicines | Umar Saidu Mohammed Auwal Ibrahim Harry P de Koning James H McKerrow Conor R Caffrey | 2023/12 | |
Coumarin-based derivatives targeting Trypanosoma cruzi cruzain and Trypanosoma brucei cathepsin L-like proteases | New Journal of Chemistry | Jéssica Alves Nunes Fabrícia Nunes da Silva Elany Barbosa da Silva Clara Andrezza Crisóstomo Bezerra Costa Johnnatan Duarte de Freitas | 2023 |
Antileishmanial compounds, compositions and use thereof | 2023/11/30 | ||
Molecular identification of phlebotomine sand flies and the harbored Leishmania spp. in Sokoto State, Nigeria | Frontiers in Cellular and Infection Microbiology | Mahmud Usman Audu Joseph Natala Isa Danladi Jatau Ndudim Isaac Ogo Ghulam Jeelani | 2023/8/31 |
The importance of good practices and false hits for QSAR-driven virtual screening real application: a SARS-CoV-2 main protease (Mpro) case study | Mateus Sá Magalhães Serafim Simone Queiroz Pantaleão Elany Barbosa da Silva James H McKerrow Anthony J O’Donoghue | 2023/7/25 | |
Structure-based discovery of thiosemicarbazones as SARS-CoV-2 main protease inhibitors | Future Medicinal Chemistry | Vinícius Gonçalves Maltarollo Elany Barbosa da Silva Thales Kronenberger Marina Mol Sena Andrade Gabriel V de Lima Marques | 2023/6 |
Discovery of pyrazolopyrrolidinones as potent, broad-spectrum inhibitors of Leishmania infection | Frontiers in tropical diseases | John A Kavouris Laura-Isobel McCall Miriam A Giardini Geraldine De Muylder Diane Thomas | 2023/1/17 |
Discovery of triple inhibitors of both SARS-CoV-2 proteases and human cathepsin L | Pharmaceuticals | Ittipat Meewan Jacob Kattoula Julius Y Kattoula Danielle Skinner Pavla Fajtová | 2022/6/13 |
Intramolecular Interactions Enhance the Potency of Gallinamide A Analogues against Trypanosoma cruzi | Journal of Medicinal Chemistry | Elany Barbosa Da Silva Vandna Sharma Lilian Hernandez-Alvarez Arthur H Tang Alexander Stoye | 2022/2/21 |
Identification of Novel Genes and Proteoforms in Angiostrongylus costaricensis through a Proteogenomic Approach | Pathogens | Esdras Matheus Gomes da Silva Karina Mastropasqua Rebello Young-Jun Choi Vitor Gregorio Alexandre Rossi Paschoal | 2022/10/31 |
Identification of Leucinostatins from Ophiocordyceps sp. as Antiparasitic Agents against Trypanosoma cruzi | ACS omega | Jean A Bernatchez Yun-Seo Kil Elany Barbosa da Silva Diane Thomas Laura-Isobel McCall | 2022/1/28 |
Anti-parasitic compounds and uses thereof | 2022/10/27 | ||
Structure-Based Identification of Naphthoquinones and Derivatives as Novel Inhibitors of Main Protease Mpro and Papain-like Protease PLpro of SARS-CoV-2 | Journal of Chemical Information and Modeling | Lucianna H Santos Thales Kronenberger Renata G Almeida Elany B Silva Rafael EO Rocha | 2022/8/12 |
Small-molecule thioesters as SARS-CoV-2 main protease inhibitors: enzyme inhibition, structure–activity relationships, antiviral activity, and X-ray structure determination | Journal of Medicinal Chemistry | Thanigaimalai Pillaiyar Philipp Flury Nadine Krüger Haixia Su Laura Schäkel | 2022/6/16 |
Dysregulation of Glycerophosphocholines in the Cutaneous Lesion Caused by Leishmania major in Experimental Murine Models | Pathogens | Adwaita R Parab Diane Thomas Sharon Lostracco-Johnson Jair L Siqueira-Neto James H McKerrow | 2021/5/13 |
Discovery of Potent Triple Inhibitors of Both SARS-CoV-2 Proteases and Human Cathepsin L | bioRxiv | Ittipat Meewan Jacob Kattoula Julius Y Kattoula Danielle Skinner Pavla Fajtová | 2021/10/20 |
Insights into the L3 to L4 developmental program through proteomics | bioRxiv | Sasisekhar Bennuru Zhaojing Meng James McKerrow Sara Lustigman Thomas B Nutman | 2021/5/6 |
Spatial metabolomics identifies localized chemical changes in heart tissue during chronic cardiac Chagas Disease | PLoS Neglected Tropical Diseases | Danya A Dean Gautham Gautham Jair L Siqueira-Neto James H McKerrow Pieter C Dorrestein | 2021/10/4 |
A clinical-stage cysteine protease inhibitor blocks SARS-CoV-2 infection of human and monkey cells | ACS chemical biology | Drake M Mellott Chien-Te Tseng Aleksandra Drelich Pavla Fajtová Bala C Chenna | 2021/3/31 |
