Hugo Gutierrez-de-Teran
Uppsala Universitet
H-index: 34
Europe-Sweden
Top articles of Hugo Gutierrez-de-Teran
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Exploring Biginelli-based scaffolds as A2B adenosine receptor antagonists: Unveiling novel structure-activity relationship trends, lead compounds, and potent colorectal … | Biomedicine & pharmacotherapy | Rubén Prieto-Díaz Hugo Fojo-Carballo Maria Majellaro Tana Tandarić Jhonny Azuaje | 2024/4/1 |
N-(Heteroaryl) thiophene sulfonamides as angiotensin AT2 receptor ligands | European Journal of Medicinal Chemistry | Johan Wannberg Johan Gising Martin Henriksson Duc Duy Vo Jonas Sävmarker | 2024/2/5 |
Visualizing the impact of disease-associated mutations on G protein–nucleotide interactions | bioRxiv | Kara Anazia Lucien Koenekoop Guillaume Ferré Enzo Petracco Hugo Gutiérrez-de-Teran | 2024 |
Discovery of allosteric modulators of A2A receptors | Tana Tandarić Hugo Gutierrez de Teran | 2023 | |
Exploring the Effect of Halogenation in a Series of Potent and Selective A2B Adenosine Receptor Antagonists | Journal of Medicinal Chemistry | Rubén Prieto-Díaz Manuel González-Gómez Hugo Fojo-Carballo Jhonny Azuaje Abdelaziz El Maatougui | 2022/12/14 |
Exploring Non-orthosteric Interactions with a Series of Potent and Selective A3 Antagonists | ACS Medicinal Chemistry Letters | Darío Miranda-Pastoriza Rodrigo Bernárdez Jhonny Azuaje Rubén Prieto-Díaz Maria Majellaro | 2022/1/10 |
A2B adenosine receptor antagonists rescue lymphocyte activity in adenosine-producing patient-derived cancer models | Journal for Immunotherapy of Cancer | Apple Hui Min Tay Rubén Prieto-Díaz Shiyong Neo Le Tong Xinsong Chen | 2022 |
Pan-cancer functional analysis of somatic mutations in G protein-coupled receptors | Scientific Reports | BJ Bongers M Gorostiola González X Wang HWT van Vlijmen Willem Jespers | 2022/12/13 |
Slow conformational dynamics of the human A2A adenosine receptor are temporally ordered | Structure | Shushu Wei Naveen Thakur Arka P Ray Beining Jin Samuel Obeng | 2022/3/3 |
Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1 Antagonists | Journal of Medicinal Chemistry | Cristina Val Carlos Rodríguez-García Rubén Prieto-Díaz Abel Crespo Jhonny Azuaje | 2022/1/22 |
Potent and Subtype-Selective Dopamine D2 Receptor Biased Partial Agonists Discovered via an Ugi-Based Approach | Journal of Medicinal Chemistry | Ana Mallo-Abreu Irene Reyes-Resina Jhonny Azuaje Rafael Franco Aitor García-Rey | 2021/6/10 |
N-(Methyloxycarbonyl) thiophene sulfonamides as high affinity AT2 receptor ligands | Bioorganic & Medicinal Chemistry | Johan Wannberg Johan Gising Jens Lindman Jessica Salander Hugo Gutiérrez-de-Terán | 2021/1/1 |
3, 4-Dihydropyrimidin-2 (1 H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure–Activity Relationship Studies, and Enantiospecific Recognition | Journal of Medicinal Chemistry | María Majellaro Willem Jespers Abel Crespo María J Núñez Silvia Novio | 2021 |
Physiological, Pathological Roles and Pharmacology of Insulin Regulated Aminopeptidase | Siew Yeen Chai Hugo Gutiérrez-de-Terán Efstratios Stratikos | 2021/4/23 | |
Deciphering conformational selectivity in the A2A adenosine G protein-coupled receptor by free energy simulations | PLOS Computational Biology | Hugo Gutierrez-de-Teran Willem Jespers Laura H. Heitman Adriaan P. IJzerman Eddy Sotelo Gerard J. P. van Westen | 2021 |
Structural basis of inhibition of human insulin-regulated aminopeptidase (IRAP) by Benzopyran-based inhibitors | ACS omega | Sudarsana Reddy Vanga Jonas Sävmarker Leelee Ng Mats Larhed Mathias Hallberg | 2018/4/25 |
Potent Inhibition of Nicotinamide N-Methyltransferase by Alkene-Linked Bisubstrate Mimics Bearing Electron Deficient Aromatics | Journal of Medicinal Chemistry | Yongzhi Gao Matthijs J Van Haren Ned Buijs Paolo Innocenti Yurui Zhang | 2021/8/23 |
Design, synthesis, HER2 inhibition and anticancer evaluation of new substituted 1, 5-dihydro-4, 1-benzoxazepines | Journal of Enzyme Inhibition and Medicinal Chemistry | Olga Cruz-López Matilde Ner Francho Nerín-Fonz Yaiza Jiménez-Martínez David Araripe | 2021/1/1 |
Identification of V6.51L as a selectivity hotspot in stereoselective A2B adenosine receptor antagonist recognition | Scientific Reports | Xuesong Wang Willem Jespers Rubén Prieto-Díaz Maria Majellaro Adriaan P IJzerman | 2021/7/8 |
Free energy calculations for protein–ligand binding prediction | Willem Jespers Johan Åqvist Hugo Gutiérrez-de-Terán | 2021 |
Co-Authors
