H.S. Overkleeft
Universiteit Leiden
H-index: 87
Europe-Netherlands
Top articles of H.S. Overkleeft
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Detection of Sulfoquinovosidase Activity in Cell Lysates Using Activity‐Based Probes | Angewandte Chemie International Edition | Zirui Li Isabelle Pickles Mahima Sharma Benjamin Melling Jeroen Codee | 2024/4/22 |
Synthesis and Macrodomain Binding of Gln‐carba‐ADPr‐peptide | ChemBioChem | Sander B Engelsma Aurelio Pio Nardozza Pieter de Saint Aulaire Herman S Overkleeft Gijsbert A van Der Marel | 2024/4/16 |
Conformational and Electronic Variations in 1, 2‐and 1, 6‐Cyclophellitols and Their Impact on Retaining α‐Glucosidase Inhibition | Chemistry–A European Journal | Tim P Ofman Jurriaan JA Heming Alba Nin-Hill Florian Küllmer Elisha Moran | 2024/3/28 |
Synthesis and application of bacterial exopolysaccharides | Gijs Ruijgrok Dung-Yeh Wu Herman S Overkleeft Jeroen DC Codée | 2024/2/1 | |
Solid‐Phase Synthesis and Biological Evaluation of Peptides ADP‐Ribosylated at Histidine | Angewandte Chemie International Edition | Hugo Minnee Johannes GM Rack Gijsbert A van der Marel Herman S Overkleeft Jeroen DC Codée | 2024/1/22 |
High-dose carfilzomib achieves superior anti-tumor activity over low-dose and recaptures response in relapsed/refractory multiple myeloma resistant to low-dose carfilzomib by … | Haematologica | Xiang Zhou Andrej Besse Jessica Peter Maximilian Johannes Steinhardt Cornelia Vogt | 2023/6/6 |
Synthetic Dual Cysteine-ADP Ribosylated Peptides from the Androgen Receptor are Recognized by the DTX3L/PARP9 Complex | ACS Chemical Biology | Sven Wijngaarden Chunsong Yang Carlos Vela-Rodríguez Lari Lehtiö Herman S Overkleeft | 2023/11/8 |
Molecular Basis for Inhibition of Heparanases and β-Glucuronidases by Siastatin B | Journal of the American Chemical Society | Yurong Chen Adrianus MCH van den Nieuwendijk Liang Wu Elisha Moran Foteini Skoulikopoulou | 2023/12/20 |
How configuration and protecting group pattern influence glycosyl acceptor reactivity | Structure-reactivity relationships in glycosylation chemistry | Jacob MA van Hengst Rik JC Hellemons Wouter A Remmerswaal Thomas Hansen Stefan van der Vorm | 2023 |
P45 HIGH-DOSE CARFILZOMIB ACHIEVES SUPERIOR ANTI-TUMOR ACTIVITY OVER LOW-DOSE AND RECAPTURES RESPONSE IN RELAPSED/REFRACTORY MULTIPLE MYELOMA RESISTANT TO LOW-DOSE CARFILZOMIB … | HemaSphere | X Zhou A Besse J Peter MJ Steinhardt C Vogt | 2023/5/1 |
β-L-Arabinofurano-cyclitol Aziridines are Cysteine-directed Broad-spectrum Inhibitors and Activity-based Probes for Retaining β-L-arabinofuranosidases | ACS Chemical Biology | Valentina Borlandelli Wendy A Offen Olga Moroz Alba Nin-Hill Nicholas McGregor | 2023/12/5 |
Activity‐Based Protein Profiling in Methicillin‐Resistant Staphylococcus aureus Reveals the Broad Reactivity of a Carmofur‐Derived Probe | ChemBioChem | Md Jalal Uddin Hermen S Overkleeft Christian S Lentz | 2023/11/2 |
Trans-cyclosulfamidate mannose-configured cyclitol allows isoform-dependent inhibition of GH47 α-d-mannosidases through a bump–hole strategy | Chemical Science | Alexandra Males Ken Kok Alba Nin-Hill Nicky de Koster Sija van den Beukel | 2023 |
Design and Synthesis of Exocyclic Cyclitol Aziridines as Potential Mechanism‐Based Glycosidase Inactivators | European Journal of Organic Chemistry | Tim P Ofman Gijsbert A van Der Marel Jeroen DC Codée Hermen S Overkleeft | 2023/4/20 |
Re-Exploring the Anthracycline Chemical Space for Better Anti-Cancer Compounds | Journal of Medicinal Chemistry | Merle A van Gelder Sabina Y van der Zanden Merijn BL Vriends Roos A Wagensveld Gijsbert A van der Marel | 2023/8/10 |
β-l-Arabinofurano-cyclitol Aziridines Are Covalent Broad-Spectrum Inhibitors and Activity-Based Probes for Retaining β-l-Arabinofuranosidases | ACS Chemical Biology | Valentina Borlandelli Wendy Offen Olga Moroz Alba Nin-Hill Nicholas McGregor | 2023/12/5 |
The development of a broad-spectrum retaining β-exo-galactosidase activity-based probe | Organic & biomolecular chemistry | Chi-Lin Kuo Qin Su Adrianus MCH van den Nieuwendijk Thomas JM Beenakker Wendy A Offen | 2023 |
4‐O‐Substituted Glucuronic Cyclophellitols are Selective Mechanism‐Based Heparanase Inhibitors | ChemMedChem | Valentina Borlandelli Zachary Armstrong Alba Nin‐Hill Jeroen DC Codée Lluís Raich | 2023/2/14 |
Four of a Kind: A Complete Collection of ADP-Ribosylated Histidine Isosteres Using Cu (I)-and Ru (II)-Catalyzed Click Chemistry | The Journal of Organic Chemistry | Hugo Minnee Hayley Chung Johannes Gregor Matthias Rack Gijsbert A van der Marel Herman S Overkleeft | 2023/7/19 |
Selection and enrichment of microbial species with an increased lignocellulolytic phenotype from a native soil microbiome by activity-based probing | ISME communications | Nicholas J Reichart Andrea K Steiger Elise M Van Fossen Ryan McClure Herman S Overkleeft | 2023/12 |
