Francesca Musumeci

Francesca Musumeci

Università degli Studi di Genova

H-index: 24

Europe-Italy

About Francesca Musumeci

Francesca Musumeci, With an exceptional h-index of 24 and a recent h-index of 21 (since 2020), a distinguished researcher at Università degli Studi di Genova, specializes in the field of medicinal chemistry.

His recent articles reflect a diverse array of research interests and contributions to the field:

Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling

Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment

Small Molecule Tyrosine Kinase Inhibitors (TKIs) for Glioblastoma Treatment

Inhibition of serum-and glucocorticoid-induced kinase 1 ameliorates hydrocephalus in preclinical models

Identification and Biological Characterization of the Pyrazolo[3,4-d]pyrimidine Derivative SI388 Active as Src Inhibitor

Virtual Screening Combined with Enzymatic Assays to Guide the Discovery of Novel SIRT2 Inhibitors

New Insights into the LANCL2-ABA Binding Mode towards the Evaluation of New LANCL Agonists

Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against …

Francesca Musumeci Information

University

Position

___

Citations(all)

1915

Citations(since 2020)

1116

Cited By

1200

hIndex(all)

24

hIndex(since 2020)

21

i10Index(all)

42

i10Index(since 2020)

37

Email

University Profile Page

Università degli Studi di Genova

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Francesca Musumeci Skills & Research Interests

medicinal chemistry

Top articles of Francesca Musumeci

Title

Journal

Author(s)

Publication Date

Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling

Molecules

Giancarlo Grossi

Naomi Scarano

Francesca Musumeci

Michele Tonelli

Evgeny Kanov

...

2024/4/11

Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment

Drug Development Research

Chiara Vagaggini

Debora Petroni

Ilaria D'Agostino

Federica Poggialini

Chiara Cavallini

...

2024/2

Small Molecule Tyrosine Kinase Inhibitors (TKIs) for Glioblastoma Treatment

Davide Frumento

Giancarlo Grossi

Marta Falesiedi

Francesca Musumeci

Anna Carbone

...

2024/1/23

Inhibition of serum-and glucocorticoid-induced kinase 1 ameliorates hydrocephalus in preclinical models

Fluids and Barriers of the CNS

Alexandra Hochstetler

Hillary Smith

Makenna Reed

Louise Hulme

Paul Territo

...

2023/8/18

Identification and Biological Characterization of the Pyrazolo[3,4-d]pyrimidine Derivative SI388 Active as Src Inhibitor

Journal of medicinal chemistry

Andrew J Culshaw

Stuart Bevan

Martin Christiansen

Prafula Copp

Andrew Davis

...

2006/1/26

Virtual Screening Combined with Enzymatic Assays to Guide the Discovery of Novel SIRT2 Inhibitors

International Journal of Molecular Sciences

Naomi Scarano

Elena Abbotto

Francesca Musumeci

Annalisa Salis

Chiara Brullo

...

2023/5/27

New Insights into the LANCL2-ABA Binding Mode towards the Evaluation of New LANCL Agonists

Pharmaceutics

Naomi Scarano

Francesco Di Palma

Nicola Origlia

Francesca Musumeci

Silvia Schenone

...

2023/12/12

Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against …

Pharmaceutics

Federica Poggialini

Chiara Vagaggini

Annalaura Brai

Claudia Pasqualini

Emmanuele Crespan

...

2023/1/30

Sweet Cherry Extract as Permeation Enhancer of Tyrosine Kinase Inhibitors: A Promising Prospective for Future Oral Anticancer Therapies

Pharmaceuticals

Federica Poggialini

Chiara Vagaggini

Annalaura Brai

Claudia Pasqualini

Anna Carbone

...

2023/10/27

Anti-Survival Effect of SI306 and Its Derivatives on Human Glioblastoma Cells

Pharmaceutics

Lorenzo Monteleone

Barbara Marengo

Francesca Musumeci

Giancarlo Grossi

Anna Carbone

...

2022/7/1

Inhibition of SGK1 ameliorates ventriculomegaly in a genetic rat model via regulation of TRPV4 in the choroid plexus

The FASEB Journal

Alexandra E Hochstetler

Hillary Smith

Makenna Reed

Louise Hulme

Nicola Perrotti

...

2022/5

Novel pyrazolo [3, 4-d] pyrimidines as dual Src/Bcr-Abl kinase inhibitors: synthesis and biological evaluation for chronic myeloid leukemia treatment

Bioorganic Chemistry

Salvatore Di Maria

Francesca Picarazzi

Mattia Mori

Annarita Cianciusi

Anna Carbone

...

2022/11/1

Synthetic heterocyclic derivatives as kinase inhibitors tested for the treatment of neuroblastoma

Francesca Musumeci

Annarita Cianciusi

Ilaria D’Agostino

Giancarlo Grossi

Anna Carbone

...

2021/11/23

Insights into RNA-dependent RNA polymerase inhibitors as antiinfluenza virus agents

Ilaria Giacchello

Francesca Musumeci

Ilaria D’Agostino

Chiara Greco

Giancarlo Grossi

...

2021/2/1

Development of Pyrazolo[3,4-d]pyrimidine Kinase Inhibitors as Potential Clinical Candidates for Glioblastoma Multiforme

ACS Medicinal Chemistry Letters

Chiara Greco

Vincenzo Taresco

Amanda K Pearce

Catherine E Vasey

Stuart Smith

...

2020/2/13

Starch/poly (glycerol-adipate) nanocomposites: A novel oral drug delivery device

Coatings

Ambra Vestri

Amanda K Pearce

Robert Cavanagh

Ioanna D Styliari

Carlos Sanders

...

2020/2/1

Synthesis and Antibacterial Evaluation of New Pyrazolo[3,4-d]pyrimidines Kinase Inhibitors

Molecules

Chiara Greco

Rosa Catania

Dario Leonardo Balacco

Vincenzo Taresco

Francesca Musumeci

...

2020/11/16

See List of Professors in Francesca Musumeci University(Università degli Studi di Genova)