Dr. Joseph M Hayes
University of Central Lancashire
H-index: 29
Europe-United Kingdom
Top articles of Dr. Joseph M Hayes
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Synthesis, In Silico and Kinetics Evaluation of N-(β-d-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(β-d-glucopyranosyl)-4(5)-arylimidazole-2 … | International Journal of Molecular Sciences | Levente Homolya Rachel T Mathomes Luca Varga Tibor Docsa László Juhász | 2024/4/23 |
Discovery of Potent Multikinase Type-II Inhibitors Targeting CDK5 in the DFG-out Inactive State with Promising Potential against Glioblastoma | Journal of Medicinal Chemistry | Zahra R Khan Philip J Welsby Izabela Stasik Joseph M Hayes | 2024/4/30 |
Multidisciplinary docking, kinetics and X-ray crystallography studies of baicalein acting as a glycogen phosphorylase inhibitor and determination of its’ potential against … | Chemico-biological interactions | Rachel T Mathomes Symeon M Koulas Ioannis Tsialtas George Stravodimos Philip J Welsby | 2023/9/1 |
In Silico-Motivated Discovery of Novel Potent Glycogen Synthase-3 Inhibitors: 1-(Alkyl/arylamino)-3H-naphtho[1,2,3-de]quinoline-2,7-dione Identified as a Scaffold … | Pharmaceuticals | Thomas D Emmerich Joseph M Hayes | 2023/4/28 |
Design and Synthesis of 3-(β-d-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential | Molecules | Sándor Kun Rachel T Mathomes Tibor Docsa László Somsák Joseph M Hayes | 2023/3/28 |
Computer-aided Design of Novel CDK5 Inhibitors; Towards New Treatments of Glioblastoma | Neuro-Oncology | Ms Zahra Khan Izabela Stasik Joseph Hayes | 2022/10 |
2-Acetamido-2-deoxy-d-glucono-1,5-lactone Sulfonylhydrazones: Synthesis and Evaluation as Inhibitors of Human OGA and HexB Enzymes | International Journal of Molecular Sciences | Mariann Kiss István Timári Teréz Barna Zuzana Mészáros Kristýna Slámová | 2022/1/18 |
The druggability of the ATP binding site of glycogen phosphorylase kinase probed by coumarin analogues | Current Research in Chemical Biology | Serafeim Alexopoulos Anastasia Gkouskou George Stravodimos Anastasia S Tsagkarakou Ioannis Tsialtas | 2022/1/1 |
Effects of Glycogen Synthase Kinase-3β (GSK3β) Inhibition in Glioblastoma Using Novel Compounds | Neuro-Oncology | Ms Klaudia Rzepecka Clare Lawrence Dima Moualla Joseph Hayes Ms Jane Alder | 2022/10 |
Evaluation of acrylamide-based molecularly imprinted polymer thin-sheets for specific protein capture—A myoglobin model | Biomedical Physics & Engineering Express | Mark V Sullivan Sarah R Dennison Joseph M Hayes Subrayal M Reddy | 2021/6/18 |
Structure-based design of potent selective nanomolar type-II inhibitors of glycogen synthase kinase-3β | Journal of Medicinal Chemistry | Matthew P Davies Rocio Benitez Concepcion Perez Sven Jakupovic Philip Welsby | 2021/1/27 |
Novel diarylamides and diarylureas with N-substitution dependent activity against medulloblastoma | European journal of medicinal chemistry | Christopher Lawson Thowaiba Babikr Ahmed Alta Georgia Moschou Vasiliki Skamnaki Theodora GA Solovou | 2021/12/5 |
Nanomolar inhibition of human OGA by 2-acetamido-2-deoxy-d-glucono-1, 5-lactone semicarbazone derivatives | European Journal of Medicinal Chemistry | Mariann Kiss Erna Szabó Boglárka Bocska Luu Thanh Sinh Conceicao Piedade Fernandes | 2021/11/5 |
Synthetic flavonoid derivatives targeting the glycogen phosphorylase inhibitor site: QM/MM-PBSA motivated synthesis of substituted 5, 7-dihydroxyflavones, crystallography, in … | Bioorganic Chemistry | Ben A Chetter Efthimios Kyriakis Daniel Barr Aikaterini G Karra Elisabeth Katsidou | 2020/9/1 |
Aromatic stacking facilitated self-assembly of ultrashort ionic complementary peptide sequence: β-sheet nanofibers with remarkable gelation and interfacial properties | Biomacromolecules | Jacek K Wychowaniec Ronak Patel James Leach Rachel Mathomes Vikesh Chhabria | 2020/5/13 |
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