Artur Mailyan
University of California, Santa Barbara
H-index: 15
North America-United States
Top articles of Artur Mailyan
Title | Journal | Author(s) | Publication Date |
|---|---|---|---|
Cbl inhibition increases the response of cytotoxic T cells to sub-optimal stimulation and drives enhanced anti-tumor responses alone or in combination with PD-1 blockade | Cancer Research | Livia Yamashiro Sachie Marubayashi Rameshwari Rayaji Anudari Battsooj Karim Mrouj | 2024/3/22 |
Inhibitors of hif-2alpha and methods of use thereof | 2023/5/25 | ||
Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2alpha | 2023/10/17 | ||
Development of a Robust and Scalable Synthetic Route for a Potent and Selective Isoindolinone PI3Kγ Inhibitor | Organic Process Research & Development | Artur K Mailyan Guillaume Mata Dillon H Miles Ehesan U Sharif Manmohan R Leleti | 2022/9/28 |
Synthesis of α-CF3-substituted γ, δ-didehydro lysine derivatives | Mendeleev Communications | Anna N Philippova Daria V Vorobyeva Tamara P Vasilyeva Artur K Mailyan Pavel S Gribanov | 2022/3/1 |
46P AB521, a clinical-stage, potent, and selective Hypoxia-Inducible Factor (HIF)-2α inhibitor, for the treatment of renal cell carcinoma | Annals of Oncology | KV Lawson KE Sivick Gauthier D Piovesan A Mailyan G Mata | 2022/3/1 |
Discovery and characterization of AB521, a novel, potent, and selective hypoxia-inducible factor (HIF)-2α inhibitor | Cancer Res. | Kenneth V Lawson Kelsey E Sivick Gauthier Artur K Mailyan Jeremy T Fournier Joel W Beatty | 2021/7/1 |
Scalable total synthesis, IP3R inhibitory activity of desmethylxestospongin B, and effect on mitochondrial function and cancer cell survival | Angewandte Chemie | Maša Podunavac Artur K Mailyan Jeffrey J Jackson Alenka Lovy Paula Farias | 2021/5/10 |
Abstract P206: AB521 potently and selectively inhibits pro-tumorigenic gene transcription by Hypoxia-Inducible Factor (HIF)-2α in vitro and in vivo | Molecular Cancer Therapeutics | Kelsey E Sivick Gauthier Dana Piovesan Soonweng Cho Kenneth V Lawson Patrick G Schweickert | 2021/12/1 |
Design, synthesis, and structure–activity relationship optimization of pyrazolopyrimidine amide inhibitors of phosphoinositide 3-kinase γ (PI3Kγ) | Chem Biol Lett | Thatikonda Narendar Reddy Adilson Beatriz RD Lopes MR Marques ED Santos | 2018 |
Discovery and Characterization of a Potent and Selective Inhibitor for Human Phosphoinositide‐3‐kinase γ | The FASEB Journal | Cesar Alejandro Meleza Ada Chen Jeremy Fournier Artur Mailyan Guillaume Mata | 2020/4 |
Discovery of potent and selective PI3Kγ inhibitors | Journal of Medicinal Chemistry | Samuel L Drew Rhiannon Thomas-Tran Joel W Beatty Jeremy Fournier Kenneth V Lawson | 2020/8/31 |
Concise Synthesis of (+)‐[13C4]‐Anatoxin‐a by Dynamic Kinetic Resolution of a Cyclic Iminium Ion | Angewandte Chemie International Edition | Jacob J Lacharity Artur K Mailyan Karen Y Chen Armen Zakarian | 2020/7/6 |
2, 3, 5-trisubstituted pyrazolo [1, 5-a] pyrimidine compounds | 2020/12/10 |
Co-Authors
