Paweł Zajdel
Uniwersytet Jagiellonski
H-index: 26
Europe-Poland
Top articles of Paweł Zajdel
Improving Activity of New Arylurea Agents against Multidrug-Resistant and Biofilm-Producing Staphylococcus epidermidis
ACS Medicinal Chemistry Letters
2024
Kamil Piska
H-Index: 10
Paweł Zajdel
H-Index: 16
Multistep Mechanochemical Synthesis of PZ-1190, a Multitarget Antipsychotic Agent
ACS Sustainable Chemistry & Engineering
2023/10/27
Paweł Zajdel
H-Index: 16
Superiority of the Triple-Acting 5-HT6R/5-HT3R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT6R Antagonist Intepirdine in Alleviation of …
Journal of Medicinal Chemistry
2023/10/5
Philippe Marin
H-Index: 7
Paweł Zajdel
H-Index: 16
Diabetic neuropathic pain improvement by inhibition of constitutive 5-HT 6 receptor activity in rats
2023/9/7
Paweł Zajdel
H-Index: 16
Philippe Marin
H-Index: 7
Synthesis, relative configuration and CB1 receptor affinity studies for a set of 1, 2, 3-triazole derivatives
Journal of Molecular Structure
2023/6/15
Tapio Nevalainen
H-Index: 10
Paweł Zajdel
H-Index: 16
Design and synthesis of novel arylurea derivatives of aryloxy (1-phenylpropyl) alicyclic diamines with antimicrobial activity against multidrug-resistant Gram-positive bacteria
European Journal of Medicinal Chemistry
2023/5/5
Discovery of SI 1/20 and SI 1/22 as Mutual Prodrugs of 5‐Fluorouracil and Imidazole‐Based Heme Oxygenase 1 Inhibitor with Improved Cytotoxicity in DU145 Prostate Cancer Cells
ChemMedChem
2023/4/17
The Constitutive Activity of Spinal 5-HT6 Receptors Contributes to Diabetic Neuropathic Pain in Rats
Biomolecules
2023/2/15
Paweł Zajdel
H-Index: 16
Philippe Marin
H-Index: 7
Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-Pyrrolo[3,2-c]quinoline Series
Molecules
2023/1/21
Philippe Marin
H-Index: 7
Paweł Zajdel
H-Index: 16
1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity
Biomolecules
2022/12/21
Philippe Marin
H-Index: 7
Paweł Zajdel
H-Index: 16
Ligand assisted CuAAC labelling and RP-HPLC analysis of zidovudine and Retrovir using propargyl-Fmoc probe
European Journal of Pharmaceutical Sciences
2022/11/1
Paweł Zajdel
H-Index: 16
New, Eco-Friendly Method for Synthesis of 3-Chlorophenyl and 1,1′-Biphenyl Piperazinylhexyl Trazodone Analogues with Dual 5-HT1A/5-HT7 Affinity and Its …
Molecules
2022/10/26
Gniewomir Latacz
H-Index: 17
Paweł Zajdel
H-Index: 16
Corrigendum to: Early 5-HT6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse (EMBO Molecular Medicine,(2020), 12, 5, 10.15252/emmm. 201910605)
EMBO Molecular Medicine
2022/9/7
Early 5‐HT6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse
EMBO Molecular Medicine
2022/9/7
Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3, 2-c] quinolines
European Journal of Medicinal Chemistry
2022/6/5
Effects of ketamine optical isomers, psilocybin, psilocin and norpsilocin on time estimation and cognition in rats
Psychopharmacology
2022/6
New N-aryl-N′-aryl-/(thio) ureido-/sulfamoylamino-derivatives of alkyl/alkylcarbamoyl piperazines: Effect of structural modifications on selectivity over 5-HT1A receptor
European Journal of Medicinal Chemistry
2022/5/5
Paweł Zajdel
H-Index: 16
Gniewomir Latacz
H-Index: 17
2-Phenyl-1H-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT6 Receptor Inverse Agonists with Cognition-Enhancing Activity
ACS Chemical Neuroscience
2021/3/11
Gniewomir Latacz
H-Index: 17
Maciej Pawłowski
H-Index: 3
Philippe Marin
H-Index: 7
Paweł Zajdel
H-Index: 16
Imidazopyridine-Based 5-HT6 Receptor Neutral Antagonists: Impact of N1-Benzyl and N1-Phenylsulfonyl Fragments on Different Receptor Conformational States
Journal of Medicinal Chemistry
2021/1/13
Philippe Marin
H-Index: 7
Paweł Zajdel
H-Index: 16
Novel mutual prodrug of 5-fluorouracil and heme oxygenase-1 inhibitor (5-FU/HO-1 hybrid): design and preliminary in vitro evaluation
Journal of Enzyme Inhibition and Medicinal Chemistry
2021/1/1
Luca Vanella
H-Index: 31
Paweł Zajdel
H-Index: 16
Rosario Pignatello
H-Index: 26
Sebastiano Intagliata
H-Index: 13
