Kowit Hengphasatporn

About Kowit Hengphasatporn

Kowit Hengphasatporn, With an exceptional h-index of 10 and a recent h-index of 10 (since 2020), a distinguished researcher at University of Tsukuba, specializes in the field of Drug discovery and design.

His recent articles reflect a diverse array of research interests and contributions to the field:

Unlocking E‐arylidene Steroid Derivatives as Promising α‐Glucosidase Inhibitors

FMO-guided design of darunavir analogs as HIV-1 protease inhibitors

Synthesis and biological evaluation of 2′-hydroxychalcone derivatives as AMPK activators

Machine learning‐guided design of potent darunavir analogs targeting HIV‐1 proteases: A computational approach for antiretroviral drug discovery

Communicationmachine Learning-Based QSAR and LB-PaCS-MD Guided Design of SARs-CoV-2 Main Protease Inhibitors (preprint)

Design of electron-donating group substituted 2-PAM analogs as antidotes for organophosphate insecticide poisoning

Regulatory Mimicry of Cyclin-Dependent Kinases by Conserved Herpesvirus Protein Kinases

Structural and thermodynamic insights into antibody light chain tetramer formation through 3D domain swapping

Kowit Hengphasatporn Information

University

Position

Center for Computational Sciences

Citations(all)

491

Citations(since 2020)

485

Cited By

141

hIndex(all)

10

hIndex(since 2020)

10

i10Index(all)

12

i10Index(since 2020)

12

Email

University Profile Page

Google Scholar

Kowit Hengphasatporn Skills & Research Interests

Drug discovery and design

Top articles of Kowit Hengphasatporn

Unlocking E‐arylidene Steroid Derivatives as Promising α‐Glucosidase Inhibitors

ChemistrySelect

2024/3/5

FMO-guided design of darunavir analogs as HIV-1 protease inhibitors

Scientific Reports

2024/2/13

Synthesis and biological evaluation of 2′-hydroxychalcone derivatives as AMPK activators

Bioorganic Chemistry

2024/2/1

Machine learning‐guided design of potent darunavir analogs targeting HIV‐1 proteases: A computational approach for antiretroviral drug discovery

Journal of Computational Chemistry

2024/1/4

Communicationmachine Learning-Based QSAR and LB-PaCS-MD Guided Design of SARs-CoV-2 Main Protease Inhibitors (preprint)

2024

Design of electron-donating group substituted 2-PAM analogs as antidotes for organophosphate insecticide poisoning

RSC advances

2023

Regulatory Mimicry of Cyclin-Dependent Kinases by Conserved Herpesvirus Protein Kinases

bioRxiv

2023

Kowit Hengphasatporn
Kowit Hengphasatporn

H-Index: 5

Yasuteru Shigeta
Yasuteru Shigeta

H-Index: 22

Structural and thermodynamic insights into antibody light chain tetramer formation through 3D domain swapping

Nature Communications

2023/12/8

The 8-bromobaicalein alleviated chikungunya-induced musculoskeletal inflammation and reduced the viral load in healthy adult mice

Emerging Microbes & Infections

2023/12/8

A sulfonamide chalcone inhibited dengue virus with a potential target at the SAM-binding site of viral methyltransferase.

Antiviral Research

2023/12/1

Structure—yeast α-glucosidase inhibitory activity relationship of 9-O-berberrubine carboxylates

Scientific Reports

2023/11/1

Identification of Promising Sulfonamide Chalcones as Inhibitors of SARS-CoV-2 3CLpro through Structure-Based Virtual Screening and Experimental Approaches

Journal of Chemical Information and Modeling

2023/8/15

Designing Potent α-Glucosidase Inhibitors: A Synthesis and QSAR Modeling Approach for Biscoumarin Derivatives

ACS omega

2023/7/11

A Structural Refinement Technique for Protein-RNA Complexes Based on a Combination of AI-based Modeling and Flexible Docking: A Study of Musashi-1 Protein

Bulletin of the Chemical Society of Japan

2023/7

X‐ray crystallographic and mutational analysis of the NylC precursor: catalytic mechanism of autocleavage and substrate hydrolysis of nylon hydrolase

The FEBS Journal

2023/7

Determination of the Association between Mesotrione Sensitivity and Conformational Change of 4-Hydroxyphenylpyruvate Dioxygenase via Free-Energy Analyses

Journal of Agricultural and Food Chemistry

2023/6/6

Sulfonylated Indeno[1,2-c]quinoline Derivatives as Potent EGFR Tyrosine Kinase Inhibitors

ACS omega

2023/5/23

In silico screening of chalcones and flavonoids as potential inhibitors against yellow head virus 3C-like protease

PeerJ

2023/4/24

The 8-bromobaicalein inhibited the replication of dengue, and Zika viruses and targeted the dengue polymerase

Scientific Reports

2023/3/25

N-Containing α-Mangostin Analogs via Smiles Rearrangement as the Promising Cytotoxic, Antitrypanosomal, and SARS-CoV-2 Main Protease Inhibitory Agents

Molecules

2023/1/22

See List of Professors in Kowit Hengphasatporn University(University of Tsukuba)