Alessio Nocentini

About Alessio Nocentini

Alessio Nocentini, With an exceptional h-index of 43 and a recent h-index of 40 (since 2020), a distinguished researcher at Università degli Studi di Firenze, specializes in the field of Medicinal Chemistry, Drug Design, Organic Chemistry, Computational Chemistry, Enzymatic Evaluation.

His recent articles reflect a diverse array of research interests and contributions to the field:

Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial …

Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains

Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases

Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors

Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma

Thiochromenocarbazole imide-based photosensitizers decorated with carbonic anhydrase inhibitors for the targeted treatment of hypoxic tumours

Design, synthesis, and carbonic anhydrase inhibition activities of Schiff bases incorporating benzenesulfonamide scaffold: Molecular docking application

3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII

Alessio Nocentini Information

University

Position

NEUROFARBA Dept.

Citations(all)

5999

Citations(since 2020)

5631

Cited By

2212

hIndex(all)

43

hIndex(since 2020)

40

i10Index(all)

165

i10Index(since 2020)

164

Email

University Profile Page

Google Scholar

Alessio Nocentini Skills & Research Interests

Medicinal Chemistry

Drug Design

Organic Chemistry

Computational Chemistry

Enzymatic Evaluation

Top articles of Alessio Nocentini

Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial …

Journal of Medicinal Chemistry

2024/3/4

Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains

International Journal of Molecular Sciences

2024/2/23

Silvia Bua
Silvia Bua

H-Index: 20

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases

Bioorganic Chemistry

2024/2/6

Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors

International Journal of Molecular Sciences

2024/1/12

Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma

Journal of Medicinal Chemistry

2024/1/11

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Thiochromenocarbazole imide-based photosensitizers decorated with carbonic anhydrase inhibitors for the targeted treatment of hypoxic tumours

Materials Advances

2024

Design, synthesis, and carbonic anhydrase inhibition activities of Schiff bases incorporating benzenesulfonamide scaffold: Molecular docking application

Saudi Pharmaceutical Journal

2023/12/1

Silvia Bua
Silvia Bua

H-Index: 20

Alessio Nocentini
Alessio Nocentini

H-Index: 28

3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII

Journal of Enzyme Inhibition and Medicinal Chemistry

2023/1/1

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Boron-containing carbonic anhydrases inhibitors

2023/11/19

1, 2, 3-Benzoxathiazine-2, 2-dioxides–effective inhibitors of human carbonic anhydrases

Journal of Enzyme Inhibition and Medicinal Chemistry

2023/1/1

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Discovery of indolinone-bearing benzenesulfonamides as new dual carbonic anhydrase and VEGFR-2 inhibitors possessing anticancer and pro-apoptotic properties

European Journal of Medicinal Chemistry

2023/11/5

Alessio Nocentini
Alessio Nocentini

H-Index: 28

4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting …

Journal of Medicinal Chemistry

2023/10/30

Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies

Bioorganic & Medicinal Chemistry

2023/10/30

Design and synthesis of 6-arylpyridine-tethered sulfonamides as novel selective inhibitors of carbonic anhydrase IX with promising antitumor features toward the human …

European Journal of Medicinal Chemistry

2023/10/5

Alessio Nocentini
Alessio Nocentini

H-Index: 28

1, 5-diaryl-1, 2, 4-triazole ureas as new SLC-0111 analogues endowed with dual carbonic anhydrase and VEGFR-2 inhibitory activities

Journal of Medicinal Chemistry

2023/7/28

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Carbonic anhydrases III and IX are new players in the crosstalk between adrenocortical carcinoma and its altered adipose microenvironment

Journal of Endocrinological Investigation

2023/7

6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography

Journal of Medicinal Chemistry

2023/6/7

Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates

Journal of Enzyme Inhibition and Medicinal Chemistry

2023/12/31

Fabrizio Carta
Fabrizio Carta

H-Index: 41

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Selective carbonic anhydrase IX and XII inhibitors based around a functionalized coumarin scaffold

Drug Development Research

2023/6

Shirisha Jonnalagadda
Shirisha Jonnalagadda

H-Index: 7

Alessio Nocentini
Alessio Nocentini

H-Index: 28

Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a …

Journal of Enzyme Inhibition and Medicinal Chemistry

2023/12/31

See List of Professors in Alessio Nocentini University(Università degli Studi di Firenze)

Co-Authors

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