Oleg Fedorov

Oleg Fedorov

University of Oxford

H-index: 66

Europe-United Kingdom

About Oleg Fedorov

Oleg Fedorov, With an exceptional h-index of 66 and a recent h-index of 46 (since 2020), a distinguished researcher at University of Oxford, specializes in the field of Chemical Biology.

His recent articles reflect a diverse array of research interests and contributions to the field:

Fluorescence assay for MERS-CoV Mpro activity measurement

Fluorescence assay for Enterovirus coxsackievirus A16 2A protease activity measurement

Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist

Imidazo [1, 2-b] pyridazines as inhibitors of DYRK kinases

Discovery of a Potent, Selective, and Cell-Active SPIN1 Inhibitor

Efficient large-scale exploration of fragment hit progression by exploiting binding-site purification of actives (B-SPA) through combining multi-step array synthesis and HT …

Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3

Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors

Oleg Fedorov Information

University

Position

___

Citations(all)

17854

Citations(since 2020)

7713

Cited By

13246

hIndex(all)

66

hIndex(since 2020)

46

i10Index(all)

123

i10Index(since 2020)

105

Email

University Profile Page

Google Scholar

Oleg Fedorov Skills & Research Interests

Chemical Biology

Top articles of Oleg Fedorov

Fluorescence assay for MERS-CoV Mpro activity measurement

2024/4/26

Oleg Fedorov
Oleg Fedorov

H-Index: 45

Fluorescence assay for Enterovirus coxsackievirus A16 2A protease activity measurement

2024/4/26

Oleg Fedorov
Oleg Fedorov

H-Index: 45

Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist

Journal of Medicinal Chemistry

2024/4/18

Imidazo [1, 2-b] pyridazines as inhibitors of DYRK kinases

European Journal of Medicinal Chemistry

2024/4/5

Oleg Fedorov
Oleg Fedorov

H-Index: 45

Simon E Ward
Simon E Ward

H-Index: 16

Discovery of a Potent, Selective, and Cell-Active SPIN1 Inhibitor

Journal of medicinal chemistry

2024/3/27

Efficient large-scale exploration of fragment hit progression by exploiting binding-site purification of actives (B-SPA) through combining multi-step array synthesis and HT …

2024/2/9

Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3

Bioorganic & Medicinal Chemistry Letters

2024/1/15

Discovery and Development Strategies for SARS-CoV-2 NSP3 Macrodomain Inhibitors

Pathogens

2023/2/15

Novel Inhibitors of MLLT1/3, a Critical Component of the Super-Elongation Complex (SEC), Target a Range of Molecularly Defined Acute Leukemias, with a Differential Profile to …

Blood

2023/11/28

Oleg Fedorov
Oleg Fedorov

H-Index: 45

Discovery of high-affinity small-molecule binders of the epigenetic reader YEATS4

Journal of medicinal chemistry

2022/12/23

EMT-like Activation in CLL Provides Novel Therapeutic Target

Blood

2022/11/15

Discovery of a potent dual SLK/STK10 inhibitor based on a maleimide scaffold

Journal of Medicinal Chemistry

2021/8/31

Discovery and characterization of selective and ligand-efficient DYRK inhibitors

Journal of Medicinal Chemistry

2021/8/3

Controlling intramolecular interactions in the design of selective, high-affinity ligands for the CREBBP bromodomain

Journal of medicinal chemistry

2021/7/13

Fragment binding to the Nsp3 macrodomain of SARS-CoV-2 identified through crystallographic screening and computational docking

Science advances

2021/4/14

COVID moonshot: open science discovery of SARS-CoV-2 main protease inhibitors by combining crowdsourcing, high-throughput experiments, computational simulations, and machine …

BioRxiv

2020/10/30

DFG-1 residue controls inhibitor binding mode and affinity, providing a basis for rational design of kinase inhibitor selectivity

Journal of medicinal chemistry

2020/8/12

Oleg Fedorov
Oleg Fedorov

H-Index: 45

Stefan Knapp
Stefan Knapp

H-Index: 69

See List of Professors in Oleg Fedorov University(University of Oxford)