Oleg Fedorov
University of Oxford
H-index: 66
Europe-United Kingdom
Top articles of Oleg Fedorov
Fluorescence assay for MERS-CoV Mpro activity measurement
2024/4/26
Oleg Fedorov
H-Index: 45
Fluorescence assay for Enterovirus coxsackievirus A16 2A protease activity measurement
2024/4/26
Oleg Fedorov
H-Index: 45
Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist
Journal of Medicinal Chemistry
2024/4/18
Imidazo [1, 2-b] pyridazines as inhibitors of DYRK kinases
European Journal of Medicinal Chemistry
2024/4/5
Oleg Fedorov
H-Index: 45
Simon E Ward
H-Index: 16
Discovery of a Potent, Selective, and Cell-Active SPIN1 Inhibitor
Journal of medicinal chemistry
2024/3/27
Efficient large-scale exploration of fragment hit progression by exploiting binding-site purification of actives (B-SPA) through combining multi-step array synthesis and HT …
2024/2/9
Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3
Bioorganic & Medicinal Chemistry Letters
2024/1/15
Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors
Science
2023/11/10
Matteo Ferla
H-Index: 8
Nir London
H-Index: 23
Frank Von Delft
H-Index: 34
James Bennett
H-Index: 12
Lennart Brewitz
H-Index: 8
Juliane Brun
H-Index: 5
Austin Clyde
H-Index: 3
Alessandro Contini
H-Index: 17
Milan Cvitkovic
H-Index: 6
Oleg Fedorov
H-Index: 45
Lori Ferrins
H-Index: 8
Richard Foster
H-Index: 6
Andre S Godoy
H-Index: 6
Michael Henry
H-Index: 27
Michelle Hill
H-Index: 6
Andrew Jajack
H-Index: 7
Lulu Kang
H-Index: 7
Peter W Kenny
H-Index: 18
Haim Levy
H-Index: 33
David Minh
H-Index: 13
Aaron Morris
H-Index: 9
Glaucius Oliva
H-Index: 22
Jin Pan
H-Index: 3
Discovery and Development Strategies for SARS-CoV-2 NSP3 Macrodomain Inhibitors
Pathogens
2023/2/15
Novel Inhibitors of MLLT1/3, a Critical Component of the Super-Elongation Complex (SEC), Target a Range of Molecularly Defined Acute Leukemias, with a Differential Profile to …
Blood
2023/11/28
Oleg Fedorov
H-Index: 45
Discovery of high-affinity small-molecule binders of the epigenetic reader YEATS4
Journal of medicinal chemistry
2022/12/23
James Bennett
H-Index: 12
Oleg Fedorov
H-Index: 45
Kilian Huber
H-Index: 3
Brigitt Raux
H-Index: 4
Andy Tsai
H-Index: 6
EMT-like Activation in CLL Provides Novel Therapeutic Target
Blood
2022/11/15
Discovery of a potent dual SLK/STK10 inhibitor based on a maleimide scaffold
Journal of Medicinal Chemistry
2021/8/31
Discovery and characterization of selective and ligand-efficient DYRK inhibitors
Journal of Medicinal Chemistry
2021/8/3
Controlling intramolecular interactions in the design of selective, high-affinity ligands for the CREBBP bromodomain
Journal of medicinal chemistry
2021/7/13
Fragment binding to the Nsp3 macrodomain of SARS-CoV-2 identified through crystallographic screening and computational docking
Science advances
2021/4/14
Open Science Discovery of Potent Non-Covalent SARS-CoV-2 Main Protease Inhibitors
BioRxiv
2020/10/30
James Bennett
H-Index: 12
Juliane Brun
H-Index: 5
Austin Clyde
H-Index: 3
Jason Cole
H-Index: 14
Alessandro Contini
H-Index: 17
Milan Cvitkovic
H-Index: 6
Oleg Fedorov
H-Index: 45
Matteo Ferla
H-Index: 8
Lori Ferrins
H-Index: 8
Richard Foster
H-Index: 6
Andre S Godoy
H-Index: 6
Michael Henry
H-Index: 27
Michelle Hill
H-Index: 6
Andrew Jajack
H-Index: 7
Lulu Kang
H-Index: 7
Peter W Kenny
H-Index: 18
Haim Levy
H-Index: 33
Nir London
H-Index: 23
David Minh
H-Index: 13
Aaron Morris
H-Index: 9
Glaucius Oliva
H-Index: 22
David Owen
H-Index: 32
Jin Pan
H-Index: 3
COVID moonshot: open science discovery of SARS-CoV-2 main protease inhibitors by combining crowdsourcing, high-throughput experiments, computational simulations, and machine …
BioRxiv
2020/10/30
DFG-1 residue controls inhibitor binding mode and affinity, providing a basis for rational design of kinase inhibitor selectivity
Journal of medicinal chemistry
2020/8/12
Oleg Fedorov
H-Index: 45
Stefan Knapp
H-Index: 69
A cell-free antibody engineering platform rapidly generates SARS-CoV-2 neutralizing antibodies (preprint)
2020
Xun Chen
H-Index: 11
Matteo Gentili
H-Index: 12
James Bennett
H-Index: 12
Juliane Brun
H-Index: 5
Austin Clyde
H-Index: 3
Jason Cole
H-Index: 14
Alessandro Contini
H-Index: 17
Milan Cvitkovic
H-Index: 6
Oleg Fedorov
H-Index: 45
Matteo Ferla
H-Index: 8
Richard Foster
H-Index: 6
Michelle Hill
H-Index: 6
Andrew Jajack
H-Index: 7
Peter W Kenny
H-Index: 18
Haim Levy
H-Index: 33
Nir London
H-Index: 23
Aaron Morris
H-Index: 9
David Owen
H-Index: 32
Jin Pan
H-Index: 3
John Spencer
H-Index: 23
Andrew Thompson
H-Index: 1
Vincent Voelz
H-Index: 19
Frank Von Delft
H-Index: 34
Matthew Wittmann
H-Index: 5
Nathan Wright
H-Index: 0